SCHEMBL7590494

SCHEMBL7590494

C#CCC(OC(CC#C)c1ccccc1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.35
HTR2A P28223 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
SLC6A4 P31645 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
TSHR P16473 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
HRH1 P35367 1/20 0.32
MTOR P42345 1/20 0.32
RAB9A P51151 1/20 0.32
GRM7 Q14831 1/20 0.32
DPP4 P27487 2/20 0.32
F2 P00734 1/20 0.32
PBRM1 Q86U86 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8975327 0.77 HTR2A (0.46) HTR2ATAAR1CHRNB2CHRNA4TSHR
SCHEMBL27504614 0.76 CYP1A2 (0.45) HTR2ACYP1A2CYP2D6
SCHEMBL7522491 0.76 PABPC1 (0.50) TSHRCYP3A4
SCHEMBL15195448 0.71 LMNA (0.52) TSHRRAB9A
SCHEMBL29936912 0.71 TRPA1 (0.41) HTR2ATAAR1SLC6A4TSHRCYP1A2
SCHEMBL3211981 0.71 HTR2A (0.36) HTR2ATAAR1TSHRCYP1A2CYP3A4
SCHEMBL16426370 0.71 HTR2A (0.36) HTR2ATAAR1TSHRCYP1A2CYP3A4
SCHEMBL610027 0.71 LMNA (0.52) TSHRRAB9A
SCHEMBL1129056 0.71 TAAR1 (0.52) TAAR1TSHRCYP1A2CYP3A4CYP2D6
SCHEMBL8535055 0.71 SCN4A (0.45) HTR2ATAAR1DPP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759915-B1 ASYMMETRIC SYNTHESIS OF CHIRAL SECONDARY ALCOHOLS CELL THERAPEUTICS INC (US) 2002-10-16 EP disclosed
US-5629423-A Asymmetric synthesis of chiral secondary alcohols CELL THERAPEUTICS, INC. (US) 1997-05-13 US disclosed
EP-0759915-A1 ASYMMETRIC SYNTHESIS OF CHIRAL SECONDARY ALCOHOLS CELL THERAPEUTICS, INC. (US) 1997-03-05 EP disclosed
WO-1995031450-A1 ASYMMETRIC SYNTHESIS OF CHIRAL SECONDARY ALCOHOLS CELL THERAPEUTICS, INC. (US) 1995-11-23 WO disclosed