SCHEMBL7591027

SCHEMBL7591027

CC#CC(C)(C)c1ccc(OC)c(C=O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.47
TSHR P16473 2/20 0.47
KDM4E B2RXH2 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 2/20 0.40
HPGD P15428 1/20 0.40
TUBB1 Q9H4B7 1/20 0.39
MAPT P10636 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PRKDC P78527 2/20 0.37
ERN1 O75460 3/20 0.36
TLR2 O60603 1/20 0.35
TLR1 Q15399 1/20 0.35
TLR6 Q9Y2C9 1/20 0.35
AOX1 Q06278 1/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
NFE2L2 Q16236 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7130351 0.85 ALDH1A1 (0.45) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL7591252 0.84 ALDH1A1 (0.44) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL7588840 0.83 ALDH1A1 (0.44) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL7587116 0.83 ALDH1A1 (0.44) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL7591439 0.82 ALDH1A1 (0.41) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL7585928 0.82 ALDH1A1 (0.41) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL4186655 0.80 ALDH1A1 (0.52) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL31738417 0.80 ALDH1A1 (0.52) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL7591958 0.78 ALDH1A1 (0.46) ALDH1A1TSHRKDM4ETDP1LMNA
SCHEMBL7616411 0.78 ALDH1A1 (0.48) ALDH1A1TSHRKDM4ETDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780375-B1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER (US) 2002-09-11 EP disclosed
US-5789423-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS; GASTROINTESTINAL AND CENTRAL NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-08-04 US disclosed
EP-0780375-A1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER INC. (US) 1997-06-25 EP disclosed