SCHEMBL7585928

SCHEMBL7585928

COC(=O)C#CC(C)(C)c1ccc(OC)c(C=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 3/20 0.41
TSHR P16473 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
ERN1 O75460 5/20 0.35
BACE1 P56817 1/20 0.35
TUBB1 Q9H4B7 1/20 0.35
TRPV1 Q8NER1 2/20 0.34
TLR2 O60603 1/20 0.34
TLR1 Q15399 1/20 0.34
TLR6 Q9Y2C9 1/20 0.34
AOX1 Q06278 1/20 0.34
JUN P05412 1/20 0.34
NFKB1 P19838 1/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7591027 0.82 ALDH1A1 (0.47) ALDH1A1KDM4ETSHRTDP1POLB
SCHEMBL7130351 0.80 ALDH1A1 (0.45) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL7591252 0.78 ALDH1A1 (0.44) ALDH1A1KDM4ETSHRTDP1POLB
SCHEMBL7588840 0.77 ALDH1A1 (0.44) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL7587116 0.77 ALDH1A1 (0.44) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL7591439 0.76 ALDH1A1 (0.41) ALDH1A1KDM4ETSHRTDP1POLB
SCHEMBL7614307 0.75 ALDH1A1 (0.48) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL4186655 0.75 ALDH1A1 (0.52) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL31738417 0.75 ALDH1A1 (0.52) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL7583554 0.75 ALDH1A1 (0.44) ALDH1A1KDM4ETSHRTDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780375-B1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER (US) 2002-09-11 EP disclosed
US-5789423-A ANTIALLERGENS, ANTIINFLAMMATORY AGENTS; GASTROINTESTINAL AND CENTRAL NERVOUS SYSTEM DISORDERS PFIZER INC. (US) 1998-08-04 US disclosed
EP-0780375-A1 3-((5-substituted benzyl)amino)-2-phenylpiperidines as substance p antagonists PFIZER INC. (US) 1997-06-25 EP disclosed