SCHEMBL7593020

SCHEMBL7593020

COc1ccc(CNc2nc3ccccc3n2-c2ncccn2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.67
LMNA P02545 2/20 0.67
SMN1; SMN2 Q16637 4/20 0.60
MAPT P10636 2/20 0.60
KMT2A Q03164 2/20 0.57
MEN1 O00255 1/20 0.57
NPC1 O15118 6/20 0.57
RAB9A P51151 6/20 0.57
THRB P10828 2/20 0.50
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
PKM P14618 1/20 0.48
GAA P10253 1/20 0.47
ALDH1A1 P00352 1/20 0.47
EGFR P00533 1/20 0.47
POLB P06746 1/20 0.47
NR2F2 P24468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11898237 0.81 LMNA (0.64) TP53LMNASMN1; SMN2MAPTKMT2A
SCHEMBL27915823 0.78 LMNA (0.77) TP53LMNASMN1; SMN2MAPTKMT2A
SCHEMBL26597943 0.77 TP53 (0.52) TP53LMNASMN1; SMN2MAPTKMT2A
SCHEMBL28806937 0.76 TP53 (0.57) TP53LMNASMN1; SMN2MAPTKMT2A
SCHEMBL28809095 0.75 TP53 (0.55) TP53LMNASMN1; SMN2MAPTKMT2A
SCHEMBL5622343 0.71 VNN1 (0.59) MAPTKMT2AMEN1NPC1RAB9A
SCHEMBL16940824 0.71 TP53 (0.50) TP53LMNASMN1; SMN2MAPTKMT2A
SCHEMBL31500073 0.71 LCK (0.61) TP53LMNASMN1; SMN2MAPTKMT2A
SCHEMBL2312890 0.69 CXCR4 (0.74) TP53MAPTKMT2ANPC1RAB9A
SCHEMBL30102083 0.69 CXCR4 (0.74) TP53MAPTKMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206265-A4 SRC KINASE INHIBITOR COMPOUNDS MERCK & CO INC (US) 2002-08-07 EP disclosed
EP-1206265-A1 SRC KINASE INHIBITOR COMPOUNDS Merck & Co., Inc. (US) 2002-05-22 EP disclosed
WO-2001000213-A1 SRC KINASE INHIBITOR COMPOUNDS MERCK & CO., INC. (US) 2001-01-04 WO disclosed