SCHEMBL75946

SCHEMBL75946

Brc1ccc(-c2cccc3c2oc2ccccc23)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.60
TNKS O95271 1/20 0.47
GGPS1 O95749 1/20 0.44
PRKDC P78527 5/20 0.43
MAOB P27338 1/20 0.41
PTGES2 Q9H7Z7 1/20 0.41
PIK3CD O00329 1/20 0.39
PIK3CB P42338 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 2/20 0.39
TSHR P16473 2/20 0.39
RAB9A P51151 2/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29403504 1.00 ALOX5 (0.60) ALOX5TNKSGGPS1PRKDCMAOB
SCHEMBL74773 0.98 ALOX5 (0.59) ALOX5TNKSGGPS1PRKDCMAOB
SCHEMBL21431985 0.95 ALOX5 (0.56) ALOX5TNKSGGPS1PRKDCMAOB
SCHEMBL28668404 0.92 ALOX5 (0.54) ALOX5TNKSGGPS1PRKDCMAOB
SCHEMBL16500881 0.91 ALOX5 (0.52) ALOX5TNKSGGPS1PRKDCMAOB
SCHEMBL12925469 0.91 ALOX5 (0.52) ALOX5TNKSGGPS1PRKDCMAOB
SCHEMBL18647422 0.91 ALOX5 (0.52) ALOX5TNKSGGPS1PRKDCMAOB
SCHEMBL16582801 0.91 ALOX5 (0.70) ALOX5GGPS1PRKDCPTGES2PIK3CD
SCHEMBL24941667 0.91 ALOX5 (0.58) ALOX5TNKSGGPS1PRKDCMAOB
SCHEMBL18022298 0.90 ALOX5 (0.51) ALOX5TNKSGGPS1PRKDCMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 792 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12588407-B2 Organic light-emitting element LG CHEM, LTD. (KR) 2026-03-24 US disclosed
US-12543495-B2 Composition, organic optoelectronic device and display device SAMSUNG SDI CO., LTD. (KR) 2026-02-03 US disclosed
US-20250234771-A1 COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENCE ELEMENT, ORGANIC ELECTROLUMINESCENCE ELEMENT, AND ELECTRONIC DEVICE IDEMITSU KOSAN CO.,LTD. (JP) 2025-07-17 US disclosed
US-20250214956-A1 ORGANIC ELECTRONIC DEVICE AND DISPLAY APPARATUS USING COMPOSITION FOR ORGANIC ELECTRONIC DEVICE DUK SAN NEOLUX CO., LTD. (KR) 2025-07-03 US disclosed
US-20250194414-A1 ARYLAMINE COMPOUND, ORGANIC ELECTROLUMINESCENCE ELEMENT AND ELECTRONIC DEVICE HODOGAYA CHEMICAL CO., LTD. (JP) 2025-06-12 US disclosed
US-12310232-B2 Composition for organic optoelectronic device, organic optoelectronic device, and display device SAMSUNG SDI CO., LTD. (KR) 2025-05-20 US disclosed
US-12289993-B2 Composition for organic optoelectronic device, organic optoelectronic device, and display device SAMSUNG SDI CO., LTD. (KR) 2025-04-29 US disclosed
US-20250129034-A1 ORGANIC COMPOUND AND ORGANIC LIGHT EMITTING DIODE COMPRISING SAME MATERIAL SCIENCE CO.,LTD. (KR) 2025-04-24 US disclosed
US-12225815-B2 Composition for organic optoelectronic device, organic optoelectronic device, and display device SAMSUNG SDI CO., LTD. (KR) 2025-02-11 US disclosed
WO-2025023719-A1 COMPOSITION FOR ORGANIC OPTOELECTRONIC DIODE, ORGANIC OPTOELECTRONIC DIODE, AND DISPLAY DEVICE 삼성에스디아이 주식회사 2025-01-30 WO disclosed
US-20060122223-A1 Substituted amino carboxylic acids THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC 2006-06-08 US disclosed
US-20060122257-A1 Phenyl substituted carboxylic acids THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC 2006-06-08 US disclosed
WO-2006055725-A2 SUBSTITUTED AMINO ACIDS AS PROTEIN TYROSINE PHOSPHATASE INHIBITORS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2006-05-26 WO disclosed
WO-2006055625-A2 HETEROCYCLYLBIPHENYL DERIVATES AS PROTEIN TYROSINE PHOSPHATASE INHIBITORS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2006-05-26 WO disclosed
EP-1622886-A2 SUBSTITUTED AMINO CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B The Institutes for Pharmaceutical Discovery, LLC (US) 2006-02-08 EP disclosed
EP-1620422-A2 PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B The Institutes for Pharmaceutical Discovery, LLC (US) 2006-02-01 EP disclosed
US-20050004369-A1 Phenyl substituted carboxylic acids INSTITUTES FOR PHARMACEUTICAL DISCOVERY, L.L.C. 2005-01-06 US disclosed
US-20040266789-A1 Substituted amino carboxylic acids INSTITUTE FOR DIABETES DISCOVERY, L.L.C. 2004-12-30 US disclosed
WO-2004099171-A2 SUBSTITUTED AMINO CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2004-11-18 WO disclosed
WO-2004099170-A2 PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2004-11-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12310232-B2 Composition for organic optoelectronic device, organic optoelectronic device, and display device OR10J3, OCIAD2, OCIAD1 ALOX5 306/4885TNKS 4526/4885GGPS1 492/4885
US-20250129034-A1 ORGANIC COMPOUND AND ORGANIC LIGHT EMITTING DIODE COMPRISING SAME SLCO4C1, SLCO2A1, OXA1L ALOX5 1660/4885TNKS 3996/4885GGPS1 1436/4885
US-20060122257-A1 Phenyl substituted carboxylic acids PTPA, PTPRS, PTPRO ALOX5 1164/4885TNKS 3446/4885GGPS1 2760/4885
US-20060122223-A1 Substituted amino carboxylic acids PTPRS, PTPRO, PTPRJ ALOX5 1550/4885TNKS 3628/4885GGPS1 2741/4885
US-20250194414-A1 ARYLAMINE COMPOUND, ORGANIC ELECTROLUMINESCENCE ELEMENT AND ELECTRONIC DEVICE SLC7A5, AHR, SLC43A1 ALOX5 412/4885TNKS 4580/4885GGPS1 4331/4885
US-12588407-B2 Organic light-emitting element LAS1L, LEF1, ARL1 ALOX5 2918/4885TNKS 3641/4885GGPS1 3410/4885
US-12225815-B2 Composition for organic optoelectronic device, organic optoelectronic device, and display device OR10J3, OCIAD2, OCIAD1 ALOX5 306/4885TNKS 4526/4885GGPS1 492/4885
US-20250214956-A1 ORGANIC ELECTRONIC DEVICE AND DISPLAY APPARATUS USING COMPOSITION FOR ORGANIC ELECTRONIC DEVICE OCIAD2, OCIAD1, EPHA4 ALOX5 2093/4885TNKS 3723/4885GGPS1 2676/4885
US-20050004369-A1 Phenyl substituted carboxylic acids PTPA, PTPRS, PTPRO ALOX5 1164/4885TNKS 3446/4885GGPS1 2760/4885
US-12543495-B2 Composition, organic optoelectronic device and display device NR2E3, OXER1, ACVRL1 ALOX5 2049/4885TNKS 3571/4885GGPS1 2197/4885
US-12289993-B2 Composition for organic optoelectronic device, organic optoelectronic device, and display device OR10J3, OCIAD2, OCIAD1 ALOX5 306/4885TNKS 4526/4885GGPS1 492/4885
US-20040266789-A1 Substituted amino carboxylic acids PTPRS, PPM1B, PTPRO ALOX5 1758/4885TNKS 3488/4885GGPS1 2583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.