SCHEMBL7595006

SCHEMBL7595006

COc1ccc([C@@H](C)N(C(=O)C(c2ccccc2)c2ccccc2)[C@H](CCCNC(=NC(=O)OCc2ccccc2)NC(=O)OCc2ccccc2)C(N)=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
ACHE P22303 2/20 0.42
ATM Q13315 1/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
BMP1 P13497 1/20 0.37
CTSL P07711 1/20 0.36
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
FOLH1 Q04609 3/20 0.36
PLAU P00749 1/20 0.36
ALOX5 P09917 1/20 0.35
ALDH1A1 P00352 3/20 0.35
CYP3A4 P08684 3/20 0.35
TSHR P16473 1/20 0.35
TP53 P04637 1/20 0.35
HDAC3 O15379 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7599024 1.00 CA1 (0.42) CA1CA2ACHEATMCNR1
SCHEMBL7601629 0.94 FOLH1 (0.40) FOLH1ALDH1A1CYP3A4TSHRKMT2A
SCHEMBL7597936 0.94 FOLH1 (0.40) FOLH1ALDH1A1CYP3A4TSHRKMT2A
SCHEMBL7600882 0.93 TRPM8 (0.41) CA1CA2ACHEHDAC1HDAC6
SCHEMBL7600478 0.93 FOLH1 (0.38) CNR1CNR2CTSLCTSSCTSK
SCHEMBL7597915 0.93 FOLH1 (0.38) CNR1CNR2CTSLCTSSCTSK
SCHEMBL7596771 0.92 CA1 (0.38) CA1CA2ACHEATMCNR1
SCHEMBL7600372 0.91 CA1 (0.39) CA1CA2ACHEATMCNR1
SCHEMBL7600355 0.90 CA1 (0.45) CA1CA2ACHEATMCNR1
SCHEMBL7597929 0.90 CA1 (0.45) CA1CA2ACHEATMCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017672-B1 NEW NPY ANTAGONISTS ASTRAZENECA AB (SE) 2002-11-27 EP disclosed