SCHEMBL7596715

SCHEMBL7596715

Cc1cc(N2CCN(CCCCC3(OC(=O)NCC(F)(F)F)c4ccccc4-c4ccccc43)CC2)nc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.43
HTR3A P46098 2/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 4/20 0.42
HPGD P15428 2/20 0.42
POLB P06746 1/20 0.42
ALOX12 P18054 1/20 0.42
DRD3 P35462 7/20 0.41
DRD2 P14416 5/20 0.41
KDM4E B2RXH2 6/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 4/20 0.40
MCHR1 Q99705 1/20 0.40
RAD52 P43351 2/20 0.40
MAPT P10636 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
ACHE P22303 1/20 0.39
HTR2A P28223 1/20 0.39
ACACB O00763 1/20 0.39
ACACA Q13085 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6776247 0.88 MTTP (0.51) HTR1AHTR3AKMT2AALDH1A1HPGD
SCHEMBL7601003 0.86 HTR1A (0.51) HTR1AHTR3ADRD3DRD2HTR2A
SCHEMBL7597136 0.86 NPC1 (0.40) HTR1AHTR3AALDH1A1HPGDDRD3
SCHEMBL7597277 0.85 HTR1A (0.49) HTR1AHTR3ADRD3DRD2HTR2A
SCHEMBL7600344 0.85 HTR3A (0.42) HTR1AHTR3ADRD3DRD2HTR2A
SCHEMBL7593152 0.85 HTR1A (0.42) HTR1AHTR3ADRD3DRD2MCHR1
SCHEMBL7720309 0.85 DRD3 (0.51) HTR1ADRD3DRD2HTR2ACHRM2
SCHEMBL7599958 0.84 DRD3 (0.43) HTR1ADRD3DRD2MCHR1CHRM2
SCHEMBL7596491 0.84 HTR1A (0.48) HTR1AHTR3ADRD3DRD2HTR2A
SCHEMBL7596831 0.83 HTR1A (0.42) HTR1ADRD3DRD2HTR2ACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255736-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) Boehringer Ingelheim Pharma KG (DE) 2002-11-13 EP disclosed
WO-2001047898-A2 SUBSTITUTED PIPERAZINE DERIVATIVES AND THEIR USE AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-07-05 WO disclosed