SCHEMBL7601983

SCHEMBL7601983

C=C(O)C(c1ccc(Cn2nc(C(F)(F)F)ccc2=O)cc1)C1CCCC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
AGTR2 P50052 1/20 0.37
HRH3 Q9Y5N1 2/20 0.37
GAA P10253 1/20 0.36
PTGS2 P35354 1/20 0.34
PTGER4 P35408 3/20 0.34
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
POLB P06746 1/20 0.33
C3AR1 Q16581 2/20 0.33
GRIA2 P42262 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PREP P48147 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1178145 0.91 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2AGTR2HRH3GAA
SCHEMBL1177948 0.83 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2AGTR2HRH3GAA
SCHEMBL7601254 0.81 POLB (0.55) ALDH1A1SMN1; SMN2HRH3CNR1CNR2
SCHEMBL7606160 0.78 PTGS2 (0.61) PTGS2
Bicarbonate SCHEMBL3692775 0.78 PTGES (0.45) ALDH1A1SMN1; SMN2PTGS2MAPT
SCHEMBL1179153 0.77 PTGES (0.58) PTGS2
SCHEMBL1178294 0.76 PTGES (0.44) ALDH1A1SMN1; SMN2PTGS2MAPT
SCHEMBL3691465 0.76 PTGS2 (0.45) PTGS2
SCHEMBL1178774 0.75 PTGS2 (0.69) PTGS2
SCHEMBL1080459 0.75 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2HRH3CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2268625-B1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF Bayer Pharma AG (DE) 2012-05-16 EP disclosed