SCHEMBL7602818

SCHEMBL7602818

CCCCCc1cccc(Cl)c1OCCN1CCN(C2=COC(C3=CC=CCC3)=CO2)CC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.36
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
DRD2 P14416 4/20 0.33
DRD3 P35462 3/20 0.33
HTR2A P28223 3/20 0.32
DRD4 P21917 1/20 0.32
HTR2C P28335 1/20 0.32
LTA4H P09960 1/20 0.31
POLB P06746 1/20 0.31
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7130569 0.87 HTR1A (0.34) HTR1AKDM4EALDH1A1
SCHEMBL7128154 0.86 HTR1A (0.42) HTR1ADRD2DRD3HTR2ADRD4
SCHEMBL7128136 0.82 ALDH1A1 (0.42) HTR1AKDM4EDRD2HTR2AALDH1A1
SCHEMBL7130709 0.79 L3MBTL1 (0.41) HTR1AKDM4EDRD2DRD3DRD4
SCHEMBL7128466 0.79 L3MBTL1 (0.47) HTR1AKDM4ELMNADRD2DRD3
SCHEMBL7124375 0.76 HTR1A (0.33) HTR1ADRD2DRD3HTR2ADRD4
SCHEMBL7126591 0.76 ALDH1A1 (0.34) HTR1ADRD2DRD3HTR2ADRD4
SCHEMBL7129896 0.76 HTR1A (0.35) HTR1AKDM4ELMNADRD2DRD3
SCHEMBL3917127 0.76 DRD2 (0.51) HTR1ADRD2HTR2AHTR2C
SCHEMBL3914428 0.76 DRD2 (0.51) HTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246820-A1 NOVEL HETEROARYL DERIVATIVES, THEIR PREPARATION AND USE H. LUNDBECK A/S (DK) 2002-10-09 EP disclosed
WO-2001049683-A1 NOVEL HETEROARYL DERIVATIVES, THEIR PREPARATION AND USE H. LUNDBECK A/S (DK) 2001-07-12 WO disclosed