SCHEMBL7605532

SCHEMBL7605532

Cc1ccc(Sc2ccc(N)cc2Cl)c(C)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 2/20 0.59
ICAM1 P05362 2/20 0.59
ITGAL P20701 2/20 0.59
PDE7A Q13946 2/20 0.56
CYP3A4 P08684 4/20 0.50
AR P10275 1/20 0.42
TSHR P16473 2/20 0.41
HAO1 Q9UJM8 1/20 0.41
ALDH1A1 P00352 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HTR1A P08908 7/20 0.40
HTR3A P46098 7/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
ADRB2 P07550 1/20 0.38
ADRB1 P08588 1/20 0.38
PTGS1 P23219 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610151 0.86 ITGB2 (0.74) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL7187676 0.83 ITGB2 (0.80) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL8310650 0.83 AR (0.60) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL6852277 0.81 PDE7A (0.79) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL7189506 0.79 ALDH1A1 (0.56) ITGB2ICAM1ITGALPDE7ACYP3A4
SCHEMBL29475022 0.79 HAO1 (0.55) ICAM1CYP3A4HAO1HTR1AHTR3A
SCHEMBL76793 0.79 HAO1 (0.55) ICAM1CYP3A4HAO1HTR1AHTR3A
SCHEMBL16269571 0.79 AR (0.51) CYP3A4ARHAO1HTR1AHTR3A
SCHEMBL20854802 0.77 PDE7A (0.52) PDE7ACYP3A4TSHRHAO1ALDH1A1
SCHEMBL15955901 0.76 PKM (0.43) PDE7ACYP3A4ARHAO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002541141-A 2002-12-03 JP claimed
EP-1165504-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2002-01-02 EP claimed
WO-2000059878-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2000-10-12 WO claimed
EP-1165504-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2002-01-02 EP disclosed
WO-2000059878-A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF ICOS CORPORATION (US) 2000-10-12 WO disclosed