SCHEMBL7607625

SCHEMBL7607625

Cc1cc(OCC(=O)O)ccc1N(C(=O)O)c1ccc2c3c([nH]c2c1)CNCC3

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.47
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
HTR7 P34969 1/20 0.47
ALOX15 P16050 2/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
THRB P10828 1/20 0.41
NFKB1 P19838 1/20 0.41
RECQL P46063 1/20 0.41
PMP22 Q01453 1/20 0.41
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 3/20 0.38
MAPT P10636 1/20 0.38
MCL1 Q07820 1/20 0.37
RAD52 P43351 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8458186 0.77 ADRA2A (0.47) NISCHADRA2AADRA2BADRA2CHTR7
SCHEMBL1875671 0.69 NISCH (0.63) NISCHADRA2AADRA2BADRA2CHTR7
SCHEMBL14924864 0.69 HSD17B10 (0.67) NISCHADRA2AADRA2BADRA2CHTR7
SCHEMBL1491307 0.67 HSD17B10 (0.67) NISCHADRA2AADRA2BADRA2CHTR7
SCHEMBL7447526 0.66 NISCH (0.47) NISCHADRA2AADRA2BADRA2CHTR7
SCHEMBL2980946 0.65 NISCH (0.67) NISCHADRA2AADRA2BADRA2CHTR7
SCHEMBL11773125 0.65 MCL1 (0.62) ALOX15TSHRHSD17B10LMNATHRB
Acetic Acid SCHEMBL30396484 0.64 NISCH (0.58) NISCHADRA2AADRA2BADRA2CHTR7
SCHEMBL2978779 0.63 LMNA (0.63) NISCHADRA2AADRA2BADRA2CHTR7
SCHEMBL11499063 0.62 NISCH (0.57) NISCHADRA2AADRA2BADRA2CHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0912182-A4 FIBRINOGEN RECEPTOR ANTAGONIST PRODRUGS MERCK & CO INC (US) 1999-12-29 EP disclosed
EP-0912182-A1 FIBRINOGEN RECEPTOR ANTAGONIST PRODRUGS Merck & Co., Inc. (US) 1999-05-06 EP disclosed
WO-1998000144-A1 FIBRINOGEN RECEPTOR ANTAGONIST PRODRUGS MERCK & CO., INC. (US) 1998-01-08 WO disclosed