SCHEMBL760770

SCHEMBL760770

CN(C)c1ccc2sc(OBOc3cc4cc(N(C)C)ccc4s3)cc2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.37
APP P05067 12/20 0.36
TERT O14746 1/20 0.36
INSR P06213 3/20 0.34
ALDH1A1 P00352 2/20 0.33
ALOX15 P16050 2/20 0.33
HSD17B10 Q99714 2/20 0.33
TSHR P16473 1/20 0.33
MAPT P10636 4/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
THRB P10828 3/20 0.33
MAPK1 P28482 3/20 0.33
RECQL P46063 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
TDP1 Q9NUW8 3/20 0.33
KDM4E B2RXH2 2/20 0.33
APAF1 O14727 2/20 0.33
GSR P00390 2/20 0.33
POLB P06746 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762071 0.74 BACE1 (0.59) CYP3A4CLK1DYRK1ADYRK1B
SCHEMBL13779418 0.73 APP (0.39) EGFRAPPTERTINSRALDH1A1
SCHEMBL23172762 0.71 APP (0.38) EGFRAPPTERTINSRALDH1A1
SCHEMBL23172965 0.70 APP (0.37) EGFRAPPTERTINSRALDH1A1
SCHEMBL1763599 0.70 AGXT (0.44) APP
SCHEMBL3195279 0.69 CYP2A6 (0.62) EGFRAPPTERTINSRALDH1A1
SCHEMBL3207769 0.69 CYP2A6 (0.53) EGFRAPPTERTINSRALDH1A1
SCHEMBL29955907 0.69 MGLL (0.53)
SCHEMBL760769 0.69 MGLL (0.53)
SCHEMBL10370593 0.67 CA2 (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120053345-A1 Indazole Compounds ABBOTT LABORATORIES (US) 2012-03-01 US disclosed
US-8008481-B2 Indazole compounds ABBVIE INC. 2011-08-30 US disclosed
US-20070282101-A1 Indazole compounds ABBVIE INC. 2007-12-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070282101-A1 Indazole compounds CYP3A43, CYP3A7, UGT1A1 EGFR 1936/4885APP 3504/4885TERT 1314/4885
US-20120053345-A1 Indazole Compounds CYP3A43, CYP3A7, UGT1A1 EGFR 1936/4885APP 3504/4885TERT 1314/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.