SCHEMBL7607722

SCHEMBL7607722

CC[Si](CC)(CC)O[C@@H](CBr)c1ccc(OCc2ccccc2)c(N(C(=O)OCc2ccccc2)S(C)(=O)=O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ACHE P22303 1/20 0.36
APP P05067 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SLC6A9 P48067 1/20 0.34
ACP1 P24666 1/20 0.33
PTPN12 Q05209 1/20 0.33
PTPN13 Q12923 1/20 0.33
SSU72 Q9NP77 1/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33
F7 P08709 1/20 0.33
F3 P13726 1/20 0.33
PRSS3 P35030 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606232 0.84 CYP19A1 (0.41) CYP19A1CA1CA2ACHEAPP
SCHEMBL7607726 0.83 CYP19A1 (0.38) CYP19A1APPNPC1HPGDRAB9A
SCHEMBL7606241 0.81 CYP19A1 (0.41) CYP19A1CA1CA2ACHEAPP
SCHEMBL7605348 0.78 CYP19A1 (0.44) CYP19A1F2F10PRSS1F7
SCHEMBL7605339 0.78 CYP19A1 (0.44) CYP19A1F2F10PRSS1F7
SCHEMBL5206971 0.77 CYP19A1 (0.47) CYP19A1ALDH1A1F2SMN1; SMN2
SCHEMBL7530567 0.75 L3MBTL1 (0.38) CYP19A1ALDH1A1
SCHEMBL7530324 0.75 L3MBTL1 (0.38) CYP19A1ALDH1A1
SCHEMBL14090693 0.75 CYP19A1 (0.39) CYP19A1ACP1PTPN12PTPN13SSU72
SCHEMBL5203737 0.75 CYP19A1 (0.47) CYP19A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed