SCHEMBL7607781

SCHEMBL7607781

COc1ccc2c(c1)S(=O)(=O)CCC(CN(C)C)=C2c1cccc(O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 3/20 0.38
HSD17B1 P14061 2/20 0.38
ESR1 P03372 3/20 0.34
STK10 O94804 1/20 0.34
GSK3B P49841 1/20 0.34
SLK Q9H2G2 1/20 0.34
CYP19A1 P11511 1/20 0.34
GALR1 P47211 1/20 0.33
ESR2 Q92731 1/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDR P35968 1/20 0.33
SLC10A2 Q12908 1/20 0.32
KDM4E B2RXH2 1/20 0.32
KCNA5 P22460 1/20 0.32
KCNH2 Q12809 1/20 0.32
MTNR1A P48039 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8006650 0.99 HSD17B2 (0.37) HSD17B2HSD17B1ESR1STK10GSK3B
SCHEMBL7611854 0.85 HSD17B1 (0.34) HSD17B2HSD17B1
SCHEMBL7615755 0.77 KDM4E (0.45) HSD17B2HSD17B1ESR1STK10GSK3B
SCHEMBL7607538 0.77 ESR1 (0.47) HSD17B2HSD17B1ESR1CYP19A1ESR2
Hydrochloric Acid SCHEMBL8020664 0.76 KDM4E (0.44) HSD17B2HSD17B1ESR1STK10GSK3B
Hydrochloric Acid SCHEMBL8016453 0.76 ESR1 (0.46) ESR1CYP19A1ESR2
SCHEMBL7607944 0.76 ESR1 (0.34) HSD17B2HSD17B1ESR1STK10GSK3B
Hydrochloric Acid SCHEMBL8016641 0.75 ESR1 (0.34) HSD17B2HSD17B1ESR1STK10GSK3B
SCHEMBL7592147 0.70 HTR7 (0.45) HSD17B2HSD17B1
SCHEMBL7588665 0.70 ESR1 (0.40) HSD17B2HSD17B1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922703-B1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds GRUENENTHAL GMBH (DE) 2002-12-04 EP disclosed
EP-0922703-A1 Substituted heterocyclic benzocycloalkenes and their use as analgesically active compounds Grünenthal GmbH (DE) 1999-06-16 EP disclosed