SCHEMBL7610102

SCHEMBL7610102

N[C@@H](Cc1ccc(-c2ccccn2)cc1)C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TPH1 P17752 11/20 0.61
SLC7A5 Q01650 2/20 0.60
DPP4 P27487 1/20 0.60
ALPI P09923 1/20 0.60
PKM P14618 1/20 0.60
PTGS1 P23219 1/20 0.60
XIAP P98170 1/20 0.60
HSD17B10 Q99714 1/20 0.48
HCAR2 Q8TDS4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610098 1.00 TPH1 (0.61) TPH1SLC7A5DPP4ALPIPKM
SCHEMBL30722996 1.00 TPH1 (0.61) TPH1SLC7A5DPP4ALPIPKM
Dl-Phenylalanine SCHEMBL27778634 0.89 SLC7A5 (0.71) TPH1SLC7A5DPP4ALPIPKM
SCHEMBL26158250 0.89 SLC7A5 (0.54) TPH1SLC7A5DPP4ALPIPKM
Tyrosine SCHEMBL27973453 0.86 SLC7A5 (0.67) TPH1SLC7A5DPP4ALPIPKM
Dl-Phenylalanine SCHEMBL28506940 0.84 SLC7A5 (0.63) TPH1SLC7A5DPP4ALPIPKM
SCHEMBL31295364 0.84 SLC7A5 (0.54) TPH1SLC7A5DPP4ALPIPKM
SCHEMBL30673627 0.84 SLC7A5 (0.54) TPH1SLC7A5DPP4ALPIPKM
SCHEMBL12273163 0.84 SLC7A5 (0.54) TPH1SLC7A5DPP4ALPIPKM
SCHEMBL29462215 0.84 SLC7A5 (0.54) TPH1SLC7A5DPP4ALPIPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230257343-A1 NOVEL AMINO ACID DERIVATIVES PEPTIDREAM INC (JP) 2023-08-17 US claimed
US-20250361274-A1 PEPTIDE AND PEPTIDE-CONTAINING AGENT PEPTIDREAM INC. (JP) 2025-11-27 US disclosed
EP-4541805-A1 PEPTIDE AND PEPTIDE-CONTAINING AGENT PeptiDream Inc. (JP) 2025-04-23 EP disclosed
WO-2025070731-A1 PEPTIDEPEPTIDE ペプチドリーム株式会社 2025-04-03 WO disclosed
WO-2025070720-A1 PEPTIDE ペプチドリーム株式会社 2025-04-03 WO disclosed
WO-2023243120-A1 PEPTIDE AND PEPTIDE-CONTAINING AGENT ペプチドリーム株式会社 2023-12-21 WO disclosed
US-20230257343-A1 NOVEL AMINO ACID DERIVATIVES PEPTIDREAM INC (JP) 2023-08-17 US disclosed
US-20230257343-A1 NOVEL AMINO ACID DERIVATIVES PEPTIDREAM INC (JP) 2023-08-17 US disclosed
US-20230257343-A1 NOVEL AMINO ACID DERIVATIVES PEPTIDREAM INC (JP) 2023-08-17 US disclosed
US-6448408-B1 CHEMICAL INTERMEDIATES IN PREPARATION OF N-MERCAPTOACYL DERIVATIVE OF PHENYLALANINE WITH PHARMALOGICAL ACTIVITY ZAMBON GROUP S.P.A. (IT) 2002-09-10 US disclosed
US-20020028946-A1 PROCESS FOR THE PREPARATION OF HETEROARYL-PHENYLALANINES ZAMBON GROUP S.P.A. (IT) 2002-03-07 US disclosed
EP-0948492-B1 PROCESS FOR THE PREPARATION OF HETEROARYL-PHENYLALANINES ZAMBON SPA (IT) 2001-07-11 EP disclosed
EP-0948492-A1 PROCESS FOR THE PREPARATION OF HETEROARYL-PHENYLALANINES ZAMBON GROUP S.p.A. (IT) 1999-10-13 EP disclosed
WO-1998028284-A1 PROCESS FOR THE PREPARATION OF HETEROARYL-PHENYLALANINES ZAMBON GROUP S.P.A. (IT) 1998-07-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250361274-A1 PEPTIDE AND PEPTIDE-CONTAINING AGENT BMP4, BMP1, BMPR2 TPH1 4441/4885SLC7A5 2541/4885DPP4 945/4885
US-20230257343-A1 NOVEL AMINO ACID DERIVATIVES DNPEP, BCAT1, ANPEP TPH1 3227/4885SLC7A5 21/4885DPP4 107/4885
US-20020028946-A1 PROCESS FOR THE PREPARATION OF HETEROARYL-PHENYLALANINES PAH, TYR, CYP2S1 TPH1 61/4885SLC7A5 51/4885DPP4 223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.