SCHEMBL7613630

SCHEMBL7613630

O=C(CNC(=O)OCc1ccccc1)Nc1ccccc1C(=O)c1ccccc1

nearest known ligand 0.75

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 5/20 0.75
HTT P42858 4/20 0.75
LMNA P02545 2/20 0.75
ALDH1A1 P00352 6/20 0.57
HPGD P15428 2/20 0.55
MAPK1 P28482 1/20 0.52
MAPT P10636 2/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
KDM1A O60341 1/20 0.50
RCOR1 Q9UKL0 1/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
POLB P06746 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPBWR1 P48145 1/20 0.48
MCHR1 Q99705 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7616103 0.90 NPSR1 (0.62) NPSR1HTTLMNAALDH1A1HPGD
SCHEMBL7617872 0.89 HTT (0.61) NPSR1HTTLMNAALDH1A1HPGD
SCHEMBL451742 0.88 LMNA (0.62) NPSR1HTTLMNAALDH1A1MAPK1
SCHEMBL7611175 0.86 NPSR1 (0.58) NPSR1HTTLMNAALDH1A1HPGD
SCHEMBL11785718 0.86 LMNA (0.77) NPSR1HTTLMNAALDH1A1MAPK1
SCHEMBL1484111 0.85 KDM4E (0.63) NPSR1HTTLMNAALDH1A1MAPK1
SCHEMBL7616469 0.83 HTT (0.55) NPSR1HTTLMNAALDH1A1HPGD
SCHEMBL25248863 0.83 HTT (0.59) NPSR1HTTLMNAALDH1A1MAPK1
SCHEMBL7609440 0.82 HTT (0.58) NPSR1HTTLMNAALDH1A1MAPK1
SCHEMBL11269680 0.80 NPSR1 (0.62) NPSR1HTTLMNAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739903-B1 CARBAMOYLMETHYLUREA DERIVATIVE SHIONOGI & CO (JP) 2002-01-23 EP disclosed
US-5739162-A ANTAGONIST FOR GASTRIN AND/OR CHOLECYSTOKININ B-NOT A-RECEPTORS; SIDE EFFECT REDUCTION; ANTIULCER AGENTS; OPIOD-ENHANCING ANALGESICS; GASTROINTESTINAL DISORDERS; ANXIOLYTIC AGENTS SHIONOGI & CO., LTD. (JP) 1998-04-14 US disclosed
EP-0739903-A1 CARBAMOYLMETHYLUREA DERIVATIVE SHIONOGI & CO., LTD. (JP) 1996-10-30 EP disclosed