SCHEMBL7617872

SCHEMBL7617872

O=C(CNC(=O)OCc1ccccc1)Nc1ccccc1C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.61
NPSR1 Q6W5P4 4/20 0.61
LMNA P02545 1/20 0.61
MGLL Q99685 1/20 0.48
ALDH1A1 P00352 6/20 0.47
HPGD P15428 2/20 0.47
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
PPARG P37231 2/20 0.45
PPARD Q03181 2/20 0.45
PPARA Q07869 2/20 0.45
NR1H4 Q96RI1 2/20 0.45
MAPK1 P28482 1/20 0.45
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
GAA P10253 1/20 0.44
KDM1A O60341 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7613630 0.89 NPSR1 (0.75) HTTNPSR1LMNAALDH1A1HPGD
SCHEMBL7616103 0.84 NPSR1 (0.62) HTTNPSR1LMNAALDH1A1HPGD
SCHEMBL27457577 0.82 ALDH1A1 (0.49) HTTNPSR1ALDH1A1HDAC3HDAC1
SCHEMBL7611175 0.81 NPSR1 (0.58) HTTNPSR1LMNAALDH1A1HPGD
SCHEMBL451742 0.80 LMNA (0.62) HTTNPSR1LMNAALDH1A1MAPK1
SCHEMBL7616469 0.78 HTT (0.55) HTTNPSR1LMNAALDH1A1HPGD
SCHEMBL1484111 0.77 KDM4E (0.63) HTTNPSR1LMNAALDH1A1MAPK1
SCHEMBL27455560 0.77 ALDH1A1 (0.52) ALDH1A1HDAC3HDAC1PPARGPPARD
SCHEMBL11785718 0.76 LMNA (0.77) HTTNPSR1LMNAALDH1A1MAPK1
Bromide SCHEMBL7611232 0.76 ALDH1A1 (0.51) ALDH1A1HDAC3HDAC1PPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739903-B1 CARBAMOYLMETHYLUREA DERIVATIVE SHIONOGI & CO (JP) 2002-01-23 EP disclosed
US-5739162-A ANTAGONIST FOR GASTRIN AND/OR CHOLECYSTOKININ B-NOT A-RECEPTORS; SIDE EFFECT REDUCTION; ANTIULCER AGENTS; OPIOD-ENHANCING ANALGESICS; GASTROINTESTINAL DISORDERS; ANXIOLYTIC AGENTS SHIONOGI & CO., LTD. (JP) 1998-04-14 US disclosed
EP-0739903-A1 CARBAMOYLMETHYLUREA DERIVATIVE SHIONOGI & CO., LTD. (JP) 1996-10-30 EP disclosed