SCHEMBL7615501

SCHEMBL7615501

CCN(C(=N)N(c1ccccc1C)C(C)C)c1cccc2c1C=CC2

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.36
TSHR P16473 1/20 0.36
CYP3A4 P08684 2/20 0.34
LMNA P02545 1/20 0.34
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7622243 0.95 TSHR (0.38) SIGMAR1TSHRCYP3A4LMNAMEN1
SCHEMBL7620405 0.88 CYP3A4 (0.41) SIGMAR1TSHRCYP3A4LMNAMEN1
SCHEMBL7614361 0.82 SIGMAR1 (0.50) SIGMAR1TSHRCYP3A4LMNAMEN1
SCHEMBL6727478 0.81 SIGMAR1 (0.47) SIGMAR1
SCHEMBL6727771 0.78 SIGMAR1 (0.44) SIGMAR1
SCHEMBL7457769 0.76 SIGMAR1 (0.41) SIGMAR1
SCHEMBL7619867 0.75 ALDH1A1 (0.36) SIGMAR1CYP3A4MEN1KMT2A
SCHEMBL6717067 0.73 SIGMAR1 (0.41) SIGMAR1TSHR
SCHEMBL7779720 0.72 HSD17B1 (0.38) SIGMAR1CYP3A4LMNA
SCHEMBL6719207 0.72 SIGMAR1 (0.49) SIGMAR1TSHRLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0517852-B1 TRI- AND TETRA-SUBSTITUTED GUANIDINES AND THEIR USE AS EXCITATORY AMINO ACID ANTAGONISTS OREGON STATE (US) 2002-07-10 EP claimed