SCHEMBL7620263

SCHEMBL7620263

Cc1cn([C@]2([SiH](c3ccccc3)c3ccccc3)O[C@H](C(O)C(C)(C)C)[C@@H](O)[C@H]2OCCO)c(=O)[nH]c1=O

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TK1 P04183 5/20 0.35
HPGD P15428 1/20 0.32
TK2 O00142 8/20 0.32
MAPK1 P28482 1/20 0.30
RNASE1 P07998 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8172947 0.91 TK1 (0.33) TK1HPGDTK2
SCHEMBL261290 0.85 TK1 (0.33) TK1HPGDTK2RNASE1
SCHEMBL7156110 0.77 TK1 (0.34) TK1HPGD
SCHEMBL313036 0.76 TK1 (0.32) TK1HPGDTK2
SCHEMBL7247157 0.76 TK1 (0.32) TK1HPGDTK2
SCHEMBL1738254 0.76 TK1 (0.31) TK1TK2
SCHEMBL8171836 0.76 TK1 (0.33) TK1
SCHEMBL9396549 0.74 RNASE1 (0.39) TK1TK2RNASE1
SCHEMBL7065023 0.72 TK1 (0.33) TK1HPGDTK2
SCHEMBL3696551 0.70 RNASE1 (0.36) TK1HPGDTK2RNASE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448080-B1 CONTACTING CELLS OR TISSUES IN VITRO WITH THE ANTISENSE OLIGONUCLEOTIDE OF THE INVENTION SO THAT EXPRESSION OF HUMAN WRN IS INHIBITED. ISIS PHARMACEUTICALS, INC. 2002-09-10 US disclosed
US-6440739-B1 POLYPEPTIDES; ANTICANCER AGENT; WOUND HEALING AGENTS ISIS PHARMACEUTICALS, INC. 2002-08-27 US disclosed
US-6440737-B1 POLYPEPTIDES ISIS PHARMACEUTICALS, INC. 2002-08-27 US disclosed
US-5985663-A AN ANTISENSE COMPOUND 8 TO 30 NUCLEOBASES IN LENGTH TARGETED TO A 5' UNTRANSLATED REGION OR 3' UNTRANSLATED REGION OF A NUCLEIC ACID ENCODING HUMAN INTERLEUKIN-15 ISIS PHARMACEUTICALS INC. (US) 1999-11-16 US disclosed