SCHEMBL7623255

SCHEMBL7623255

C[C@@H]1CN([C@@H](c2cccnc2)c2cccc(O)c2S(=O)(=O)C(F)(F)F)[C@@H](C)CN1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 1/20 0.35
MGLL Q99685 1/20 0.35
ABHD6 Q9BV23 1/20 0.35
CYP3A4 P08684 10/20 0.35
CYP3A5 P20815 9/20 0.35
CYP2D6 P10635 1/20 0.31
NFKB1 P19838 1/20 0.31
PRKD3 O94806 1/20 0.31
PRKCG P05129 1/20 0.31
PRKCB P05771 1/20 0.31
PRKCA P17252 1/20 0.31
PRKCH P24723 1/20 0.31
PRKCI P41743 1/20 0.31
PRKCE Q02156 1/20 0.31
PRKCQ Q04759 1/20 0.31
PRKCZ Q05513 1/20 0.31
PRKCD Q05655 1/20 0.31
PRKD1 Q15139 1/20 0.31
ADRB3 P13945 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7616431 0.81 OPRD1 (0.48) CYP3A4KDM4E
SCHEMBL7623262 0.77 MGLL (0.35) PLA2G7MGLLABHD6CYP3A4CYP3A5
SCHEMBL6526001 0.64 SIGMAR1 (0.37) CYP3A4
SCHEMBL6525998 0.64 SIGMAR1 (0.37) CYP3A4
SCHEMBL16456516 0.64 SIGMAR1 (0.37) CYP3A4
SCHEMBL15080471 0.64 SIGMAR1 (0.37) CYP3A4
SCHEMBL4576003 0.63 OPRD1 (0.43) CYP3A4CYP2D6NFKB1MAPT
SCHEMBL4499828 0.63 SIGMAR1 (0.52) CYP2D6
SCHEMBL12016528 0.62 OPRD1 (0.45)
SCHEMBL6932627 0.61 SIGMAR1 (0.43) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020052007-A1 Diarylmethylbenzylpiperazines and corresponding halobenzyl derivatives ENTA HOLDING LLC 2002-05-02 US disclosed