SCHEMBL7623262

SCHEMBL7623262

C[C@@H]1CN([C@H](c2cccnc2)c2cccc(OS(=O)(=O)C(F)(F)F)c2)[C@@H](C)CN1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.35
PLA2G7 Q13093 1/20 0.35
ABHD6 Q9BV23 1/20 0.35
CYP3A4 P08684 3/20 0.35
CYP3A5 P20815 2/20 0.35
DRD2 P14416 1/20 0.35
DRD1 P21728 1/20 0.35
DRD4 P21917 1/20 0.35
DRD5 P21918 1/20 0.35
DRD3 P35462 1/20 0.35
OPRD1 P41143 1/20 0.33
CYP19A1 P11511 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
CYP2D6 P10635 1/20 0.33
NFKB1 P19838 1/20 0.33
PRKD3 O94806 1/20 0.33
PRKCG P05129 1/20 0.33
PRKCB P05771 1/20 0.33
PRKCA P17252 1/20 0.33
PRKCH P24723 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12016528 0.83 OPRD1 (0.45) OPRD1
SCHEMBL7616455 0.81 OPRD1 (0.56) CYP3A4OPRD1CYP2D6NFKB1
SCHEMBL4576560 0.79 OPRD1 (0.50) CYP3A4OPRD1CYP2D6NFKB1
SCHEMBL4576004 0.78 OPRD1 (0.56) CYP3A4OPRD1CYP2D6NFKB1
SCHEMBL12018158 0.78 OPRD1 (0.56) CYP3A4OPRD1CYP2D6NFKB1
SCHEMBL7623255 0.77 PLA2G7 (0.35) MGLLPLA2G7ABHD6CYP3A4CYP3A5
SCHEMBL16456532 0.76 OPRD1 (0.51) OPRD1
SCHEMBL6466974 0.76 OPRD1 (0.51) OPRD1
SCHEMBL4576003 0.75 OPRD1 (0.43) CYP3A4OPRD1CYP2D6NFKB1
SCHEMBL6466971 0.73 OPRD1 (0.40) OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020052007-A1 Diarylmethylbenzylpiperazines and corresponding halobenzyl derivatives ENTA HOLDING LLC 2002-05-02 US disclosed