SCHEMBL7627010

SCHEMBL7627010

O[C@@H]1[C@H](O)[C@@H](CF)O[C@H]1n1cnc2c(NOCc3ccccc3)nc(Cl)nc21

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.60
ADORA1 P30542 4/20 0.59
ADORA2A P29274 2/20 0.59
NT5E P21589 6/20 0.59
ADORA2B P29275 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7627041 1.00 ADORA3 (0.60) ADORA3ADORA1ADORA2ANT5EADORA2B
SCHEMBL8820534 0.92 ADORA1 (0.70) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL8820548 0.92 ADORA1 (0.70) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL8820284 0.84 ALDH1A1 (0.55) ADORA3ADORA1ADORA2ANT5E
SCHEMBL8819342 0.84 ALDH1A1 (0.55) ADORA3ADORA1ADORA2ANT5E
SCHEMBL8820255 0.83 ADORA1 (0.73) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL8820273 0.83 ADORA1 (0.73) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL5353431 0.81 ADORA3 (0.67) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL8820021 0.80 ADORA1 (0.63) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL8820039 0.80 ADORA1 (0.63) ADORA3ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6455510-B1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2002-09-24 US claimed
US-5589467-A TREATING CENTRAL NERVOUS SYSTEM DISORDERS NOVO NORDISK A/S (DK) 1996-12-31 US claimed
WO-1997033590-A1 A METHOD OF TREATING DISORDERS RELATED TO CYTOKINES IN MAMMALS NOVO NORDISK A/S (DK) 1997-09-18 WO disclosed
WO-1997033591-A1 A METHOD OF TREATING DISORDERS RELATED TO CYTOKINES IN MAMMALS NOVO NORDISK A/S (DK) 1997-09-18 WO disclosed
US-5589467-A TREATING CENTRAL NERVOUS SYSTEM DISORDERS NOVO NORDISK A/S (DK) 1996-12-31 US disclosed