SCHEMBL7632279

SCHEMBL7632279

COc1ccc(C#C[Si](C)(C)C)cc1C(C)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 1/20 0.42
LMNA P02545 3/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTT P42858 3/20 0.41
PDE4A P27815 2/20 0.40
SRC P12931 1/20 0.40
TGFBR1 P36897 1/20 0.40
MAPT P10636 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
RECQL P46063 1/20 0.37
GAA P10253 1/20 0.37
GABRA1 P14867 2/20 0.37
GABRG2 P18507 2/20 0.37
GABRB3 P28472 2/20 0.37
GABRA5 P31644 2/20 0.37
GABRA3 P34903 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7634542 0.81 MAPT (0.52) LMNAALDH1A1KDM4EHSD17B10HTT
SCHEMBL18097559 0.79 GRM5 (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL30468153 0.79 AR (0.50) CA9LMNAALDH1A1KDM4EHSD17B10
SCHEMBL7632890 0.79 HTT (0.44) CA9LMNAALDH1A1KDM4EHSD17B10
SCHEMBL20855586 0.79 AR (0.50) CA9LMNAALDH1A1KDM4EHSD17B10
SCHEMBL29582057 0.78 CA2 (0.43) CA9ALDH1A1PDE4AACACB
SCHEMBL26926326 0.78 CA2 (0.43) CA9ALDH1A1PDE4AACACB
SCHEMBL5880802 0.78 GABRA1 (0.38) LMNAALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL4634208 0.77 LMNA (0.39) LMNAALDH1A1KDM4EHTTMAPT
SCHEMBL7627294 0.77 ALDH1A1 (0.52) CA9LMNAALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975573-B1 TRISUBSTITUTED PHENYL DERIVATIVES HAVING RETINOID AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE BIOLOGICAL ACTIVITY ALLERGAN SALES INC (US) 2002-09-18 EP disclosed
US-6235923-B1 RETINOIDS AND CELL DIFFERENTIATION ALLERGAN SALES, INC. 2001-05-22 US disclosed
US-6225494-B1 TREATING SKIN DISORDERS, REDUCED SIDE EFFECTS ALLERGAN SALES, INC. 2001-05-01 US disclosed
US-6037488-A COMPOUNDS SUCH AS 4-((4'-ISOPROPOXY-3'-(1-M-TOLYL)VINYL)PHENYLETHYNYL)BENZOIC ACID ALLERGAN SALES, INC. (US) 2000-03-14 US disclosed
EP-0975573-A1 TRISUBSTITUTED PHENYL DERIVATIVES HAVING RETINOID AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 2000-02-02 EP disclosed
WO-1998047854-A1 TRISUBSTITUTED PHENYL DERIVATIVES HAVING RETINOID AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1998-10-29 WO disclosed