SCHEMBL762546

SCHEMBL762546

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](C)Cc3ccc4ccccc4c3)C2)nc2c(C)cccc21

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.37
NPY1R P25929 3/20 0.36
HRH1 P35367 3/20 0.36
CYP2D6 P10635 3/20 0.36
HTR4 Q13639 3/20 0.35
TNKS O95271 3/20 0.35
PARP1 P09874 3/20 0.35
TNKS2 Q9H2K2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
TSHR P16473 2/20 0.35
KMT2A Q03164 2/20 0.35
CHRM1 P11229 1/20 0.35
CNR2 P34972 1/20 0.35
PPARA Q07869 1/20 0.34
CYP3A4 P08684 2/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739273 0.92 NPY1R (0.36) KCNH2NPY1RHRH1CYP2D6HTR4
SCHEMBL739272 0.92 NPY1R (0.36) KCNH2NPY1RHRH1CYP2D6HTR4
SCHEMBL762543 0.92 CYP2D6 (0.36) KCNH2NPY1RHRH1CYP2D6TNKS
SCHEMBL741747 0.87 HRH1 (0.36) KCNH2NPY1RHRH1CYP2D6HTR4
SCHEMBL10293031 0.87 PADI4 (0.38) KCNH2NPY1RHRH1CYP2D6ALDH1A1
SCHEMBL763304 0.84 ALDH1A1 (0.35) KCNH2HRH1CYP2D6ALDH1A1TSHR
SCHEMBL738775 0.84 CFD (0.38) KCNH2HRH1CYP2D6ALDH1A1TSHR
SCHEMBL738776 0.84 CFD (0.38) KCNH2HRH1CYP2D6ALDH1A1TSHR
SCHEMBL738703 0.84 TACR1 (0.36) KCNH2HRH1CYP2D6ALDH1A1TSHR
SCHEMBL762831 0.84 TLR8 (0.36) KCNH2NPY1RHRH1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed