SCHEMBL7635227

SCHEMBL7635227

N#Cc1nc(-c2cccnc2)nn1-c1ccc(NCC2Cc3ccccc3C2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.39
CHRNA5 P30532 2/20 0.39
CHRNA4 P43681 2/20 0.39
PDE5A O76074 2/20 0.38
GBA1 P04062 7/20 0.37
ABCG2 Q9UNQ0 2/20 0.35
ADORA2A P29274 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ADORA1 P30542 1/20 0.33
KMT2A Q03164 2/20 0.33
KDM6B O15054 1/20 0.33
NR1I2 O75469 1/20 0.33
CHRNA1 P02708 1/20 0.33
MAOB P27338 1/20 0.33
OPRM1 P35372 1/20 0.33
AHR P35869 1/20 0.33
AVPR1A P37288 1/20 0.33
OPRK1 P41145 1/20 0.33
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7632588 0.84 HDAC1 (0.39) PDE5AGBA1RAB9AKMT2AEPHX2
SCHEMBL7234847 0.81 KDM4E (0.46) CHRNB2CHRNA5CHRNA4PDE5AEPHX2
SCHEMBL7236687 0.81 PTGS2 (0.37) CHRNB2CHRNA5CHRNA4PDE5AGBA1
SCHEMBL7634848 0.77 MAPT (0.38) CHRNB2CHRNA5CHRNA4ABCG2ADORA2A
SCHEMBL7240009 0.74 EPHX2 (0.59) EPHX2
SCHEMBL7627296 0.74 MAPT (0.36) CHRNB2CHRNA5CHRNA4KMT2AMAPK1
SCHEMBL7638011 0.73 MAPT (0.45) CHRNB2CHRNA5CHRNA4KMT2AMAPK1
SCHEMBL7635766 0.71 CACNA1B (0.41) KMT2AMAPK1
SCHEMBL7244587 0.70 VCP (0.37) PDE5AGBA1EPHX2
SCHEMBL7630028 0.70 ABCB1 (0.36) ABCG2KMT2AABCB1ABCC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451820-B1 Substituted 1-(4-aminophenly)triazoles and their use as anti-inflammatory agents BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-09-17 US claimed
WO-2001072740-A1 SUBSTITUTED 1-(4-AMINOPHENYL) TRIAZOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-10-04 WO claimed