SCHEMBL7634848

SCHEMBL7634848

Cc1cccc(C)c1CNc1ccc(-n2nc(-c3cccnc3)nc2C#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.38
HDAC1 Q13547 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNA5 P30532 2/20 0.38
CHRNA4 P43681 2/20 0.38
THRB P10828 2/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 2/20 0.36
EPHX2 P34913 1/20 0.36
HPGD P15428 2/20 0.35
TSHR P16473 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
AHR P35869 1/20 0.35
RAB9A P51151 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C19 P33261 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7627296 0.94 MAPT (0.36) MAPTHDAC1HDAC6CHRNB2CHRNA5
SCHEMBL7638011 0.84 MAPT (0.45) MAPTHDAC1HDAC6CHRNB2CHRNA5
SCHEMBL7244506 0.80 PTGS2 (0.42) HDAC1HDAC6KMT2AALDH1A1HPGD
SCHEMBL7243350 0.80 ALDH1A1 (0.46) MAPTMAPK1KMT2AALDH1A1EPHX2
SCHEMBL7630672 0.78 HDAC1 (0.42) MAPTHDAC1HDAC6THRBEPHX2
SCHEMBL7635227 0.77 CHRNB2 (0.39) CHRNB2CHRNA5CHRNA4MAPK1KMT2A
SCHEMBL7243090 0.77 EPHX2 (0.42) MAPTMAPK1KMT2AALDH1A1EPHX2
SCHEMBL7243590 0.77 PTGS2 (0.39) MAPTKMT2AALDH1A1KDM4ERAB9A
SCHEMBL7635766 0.77 CACNA1B (0.41) MAPTMAPK1KMT2AALDH1A1TSHR
SCHEMBL7630028 0.75 ABCB1 (0.36) MAPTMAPK1KMT2AALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451820-B1 Substituted 1-(4-aminophenly)triazoles and their use as anti-inflammatory agents BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 2002-09-17 US claimed
WO-2001072740-A1 SUBSTITUTED 1-(4-AMINOPHENYL) TRIAZOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-10-04 WO claimed