SCHEMBL7637232

SCHEMBL7637232

c1cc(-c2nc3ccccc3[nH]2)cc(N2CC[N]CC2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.58
NPC1 O15118 6/20 0.58
RAB9A P51151 6/20 0.58
ALDH1A1 P00352 6/20 0.58
KDM4E B2RXH2 5/20 0.58
HPGD P15428 3/20 0.58
HSD17B10 Q99714 3/20 0.58
TP53 P04637 2/20 0.58
NPBWR1 P48145 1/20 0.54
GAA P10253 1/20 0.53
BACE1 P56817 2/20 0.52
ACHE P22303 1/20 0.51
DRD2 P14416 3/20 0.48
DRD3 P35462 2/20 0.48
POLB P06746 2/20 0.48
BACE2 Q9Y5Z0 1/20 0.47
PIM1 P11309 1/20 0.47
PIM3 Q86V86 1/20 0.47
AURKB Q96GD4 1/20 0.47
MEN1 O00255 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3511276 0.86 HTR7 (0.57) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL16328113 0.85 KDM4E (0.56) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL13033551 0.84 NPC1 (0.54) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL13033512 0.83 ACHE (0.76) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL13033499 0.81 KDM4E (0.55) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL3511121 0.81 DRD2 (0.58) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL13033489 0.81 ACHE (0.56) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL13033508 0.80 ACHE (0.58) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL13033513 0.80 ACHE (0.56) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL13033498 0.78 LMNA (0.64) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1210340-A1 SUBSTITUTED PIPERAZINE DERIVATIVES, THE PRODUCTION THEREOF AND THEIR UTILIZATION AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 2002-06-05 EP disclosed
WO-2001014355-A1 SUBSTITUTED PIPERAZINE DERIVATIVES, THE PRODUCTION THEREOF AND THEIR UTILIZATION AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-03-01 WO disclosed