SCHEMBL76377

SCHEMBL76377

COc1ccc(CC(=O)Cl)cc1OC

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.59
HTT P42858 3/20 0.59
NPC1 O15118 1/20 0.59
GAA P10253 5/20 0.58
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58
MAPT P10636 1/20 0.58
HPGD P15428 1/20 0.58
ALDH1A1 P00352 3/20 0.57
LDHA P00338 1/20 0.57
CA2 P00918 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.56
NPSR1 Q6W5P4 1/20 0.55
MAPK1 P28482 1/20 0.55
EPHX2 P34913 1/20 0.55
CA5A P35218 1/20 0.54
TSHR P16473 1/20 0.53
NFKB1 P19838 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
CA1 P00915 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9808605 0.89 PTGS1 (0.62) LMNAHTTNPC1GAAKMT2A
SCHEMBL2392519 0.87 LDHA (0.49) LMNAHTTNPC1GAAKMT2A
SCHEMBL18648672 0.86 CYP3A4 (0.50) LMNAHTTNPC1GAAKMT2A
SCHEMBL2391312 0.86 TSHR (0.73) LMNAGAAALDH1A1MAPK1TSHR
SCHEMBL3616256 0.86 ALDH1A1 (0.53) LMNAHTTNPC1GAAKMT2A
SCHEMBL3659918 0.86 GAA (0.50) LMNAHTTNPC1GAAKMT2A
SCHEMBL30859524 0.85 LMNA (0.63) LMNAHTTNPC1GAAKMT2A
SCHEMBL11187045 0.85 LMNA (0.63) LMNAHTTNPC1GAAKMT2A
SCHEMBL17709374 0.85 REN (0.49) LMNAHTTNPC1GAAKMT2A
SCHEMBL11281357 0.84 PTGS1 (0.53) LMNAHTTNPC1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 428 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117024298-A Tertiary amide compound containing naphthyl and its preparation method and application 北京中医药大学 2023-11-10 CN claimed
WO-2023086696-A2 APPARATUS AND METHODS FOR CONTINUOUS FLOW SYNTHESIS OF CISATRACURIUM ODH IP Corp. (US) 2023-05-19 WO claimed
CN-104829470-B One is combined into the midbody compound of Ivabradine and its application 江苏宇田医药有限公司 2017-08-25 CN claimed
CN-104829470-A Set of intermediate compounds used for synthesis of Ivabradine, and applications thereof JIANGSU YUTIAN PHARMACEUTICAL TECHNOLOGY CO LTD 2015-08-12 CN claimed
CN-102924318-B L-leucine derivatives blocking entrance of H5N1 avian influenza virus and preparation method for same UNIV WUHAN 2014-06-04 CN claimed
CN-102924318-A L-leucine derivatives blocking entrance of H5N1 avian influenza virus and preparation method for same UNIV WUHAN 2013-02-13 CN claimed
CN-101643465-A Preparation method of COMT inhibitor 5, 6, 7, 3', 4'-pentamethoxyl isoflavone UNIV DONGHUA 2010-02-10 CN claimed
EP-4582423-A1 NOVEL TRICYCLIC DERIVATIVE COMPOUND AND USES THEREOF Hanmi Pharm. Co., Ltd. (KR) 2025-07-09 EP disclosed
CN-120077041-A Tricyclic derivative compounds and use thereof 韩美药品株式会社 2025-05-30 CN disclosed
CN-118027395-B Coating material, preparation method and application thereof, and lithium battery diaphragm 安徽壹石通材料科学研究院有限公司 2025-04-29 CN disclosed
US-20250066378-A1 SPIRO-OXAZOLONES HOFFMANN-LA ROCHE INC. (US) 2025-02-27 US disclosed
US-12162887-B2 Spiro-oxazolones HOFFMANN-LA ROCHE INC. (US) 2024-12-10 US disclosed
CN-118027395-A Coating material, preparation method and application thereof, and lithium battery diaphragm 安徽壹石通材料科学研究院有限公司 2024-05-14 CN disclosed
US-4232014-A AMIDOALKYLINDANS MARION LABORATORIES, INC. (US) 1980-11-04 US disclosed
US-4191770-A ANTIULCER AGENTS, ANTISECRETORY AGENTS KALI-CHEMIE PHARMA GMBH (DE) 1980-03-04 US disclosed
US-4181738-A DOPAMINERGIC CORNELL RESEARCH FOUNDATION, INC. (US) 1980-01-01 US disclosed
US-4171370-A Phenoxy-amino-propanols MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-10-16 US disclosed
US-3962254-A HYPOTENSIVE AGENTS MARION LABORATORIES, INC. (US) 1976-06-08 US disclosed
US-3954774-A HYPOTENSIVE AGENTS MARION LABORATORIES, INC. (US) 1976-05-04 US disclosed
US-3950236-A OXIDATION, ALKYL-ALKOXY-BIBENZYL COMPOUNDS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF HEALTH, EDUCATION AND WELFARE (US) 1976-04-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12162887-B2 Spiro-oxazolones AVPR1A, AVPR1B, AVPR2 LMNA 3114/4885HTT 1513/4885NPC1 3185/4885
US-20250066378-A1 SPIRO-OXAZOLONES AVPR1A, AVPR1B, AVPR2 LMNA 3114/4885HTT 1513/4885NPC1 3185/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.