SCHEMBL7645535

SCHEMBL7645535

COc1ccc(N(CCN(CC(=O)O)C(=O)Cn2ccnc2)C(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
HMOX2 P30519 1/20 0.42
CYP19A1 P11511 4/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 2/20 0.39
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
AHR P35869 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7637174 0.93 CYP3A4 (0.47) CYP3A4CYP2D6HMOX2CYP19A1ALDH1A1
SCHEMBL9225377 0.84 IDH1 (0.45) ALDH1A1NPSR1
SCHEMBL7644923 0.84 CYP19A1 (0.38) CYP19A1ALDH1A1NPSR1
SCHEMBL7645531 0.81 CYP3A4 (0.49) CYP3A4CYP2D6HMOX2CYP19A1ALDH1A1
SCHEMBL3927370 0.77 CA12 (0.41) MAPK1
SCHEMBL7641484 0.77 CYP19A1 (0.37) CYP19A1ALDH1A1MAPK1NPSR1
SCHEMBL7641427 0.77 IDH1 (0.44) ALDH1A1KDM4ENPSR1
SCHEMBL7645537 0.76 CYP19A1 (0.44) CYP19A1ALDH1A1GAAMAPK1L3MBTL1
SCHEMBL7637169 0.76 CYP3A4 (0.48) CYP3A4CYP2D6HMOX2CYP19A1ALDH1A1
SCHEMBL7637993 0.73 MEN1 (0.48) ALDH1A1GAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7258222-A None JP disclosed
US-6465650-B1 INTERMEDIATE STEPS IN PREPARING PEPTIDE NUCLEIC ACIDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-10-15 US disclosed
US-6075143-A USEFUL FOR FORMING PEPTIDE NUCLEIC ACIDS OR HYBRID OF PEPTIDE NUCLEIC ACIDS AND DEOXYNUCLEIC ACID HOECHST AKTIENGESELLSCHAFT (DE) 2000-06-13 US disclosed
JP-H07258222-A SUBSTITUTED N-ETHYLGLYCINE DERIVATIVE FOR PRODUCING PNA AND PNA/DNA HYBRID HOECHST AG 1995-10-09 JP disclosed
EP-0672661-A1 Substituted N-ethyl-glycinderivatives for the preparation of PNA and PNA-/DNA hybrides HOECHST AKTIENGESELLSCHAFT (DE) 1995-09-20 EP disclosed