SCHEMBL7649189

SCHEMBL7649189

O=c1c2ccccc2[nH]c(=S)n1CCN1CCC(c2c[nH]c3ccccc23)CC1

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.67
ALDH1A1 P00352 1/20 0.67
KMT2A Q03164 2/20 0.66
MPO P05164 1/20 0.66
SMN1; SMN2 Q16637 1/20 0.64
HTR2A P28223 2/20 0.59
CYP2D6 P10635 2/20 0.59
CYP1A2 P05177 1/20 0.59
CYP3A4 P08684 1/20 0.59
HTR1A P08908 1/20 0.59
CYP2C9 P11712 1/20 0.59
DRD2 P14416 1/20 0.59
HPGD P15428 1/20 0.59
TSHR P16473 1/20 0.59
HTR2C P28335 1/20 0.59
ADRA1D P25100 3/20 0.58
MEN1 O00255 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11007868 0.89 ADRA1D (0.61) ALDH1A1KMT2AHTR2ACYP2D6CYP1A2
SCHEMBL14306777 0.83 ADRA1D (0.80) KDM4ECYP2D6ADRA1D
SCHEMBL2730275 0.81 ALDH1A1 (1.00) KDM4EALDH1A1KMT2AMPOSMN1; SMN2
SCHEMBL11047479 0.80 ADRA1D (0.61) HTR2ACYP2D6ADRA1D
Hydrochloric Acid SCHEMBL2730111 0.80 ALDH1A1 (0.97) KDM4EALDH1A1KMT2AMPOSMN1; SMN2
SCHEMBL2732924 0.80 KMT2A (1.00) KDM4EALDH1A1KMT2AMPOSMN1; SMN2
SCHEMBL10740720 0.80 CYP2D6 (0.53) ALDH1A1KMT2AHTR2ACYP2D6CYP1A2
SCHEMBL10744006 0.80 SLC6A4 (0.53) CYP2D6HTR1ADRD2ADRA1D
SCHEMBL11013197 0.80 DRD2 (0.61) KDM4EALDH1A1KMT2AHTR2ACYP2D6
SCHEMBL15613370 0.79 KDM4E (0.81) KDM4EALDH1A1KMT2AMPOSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492364-B1 Triazolo and derivatives as chemokine inhibitors TORAY INDUSTRIES, INC. (JP) 2002-12-10 US disclosed
EP-1067130-A1 TRIAZOLO DERIVATIVES AND CHEMOKINE INHIBITORS CONTAINING THE SAME AS THE ACTIVE INGREDIENT TORAY INDUSTRIES, INC. (JP) 2001-01-10 EP disclosed