SCHEMBL10740720

SCHEMBL10740720

O=c1[nH]c2ccc(O)cc2c(=O)n1CCN1CCC(c2c[nH]c3ccccc23)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.53
CYP1A2 P05177 2/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2C9 P11712 2/20 0.53
THPO P40225 1/20 0.53
ADRA1D P25100 4/20 0.53
SLC6A4 P31645 2/20 0.51
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
HTR1A P08908 1/20 0.51
MAPT P10636 1/20 0.51
DRD2 P14416 1/20 0.51
HPGD P15428 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
DRD1 P21728 1/20 0.51
DRD4 P21917 1/20 0.51
HTR1D P28221 1/20 0.51
HTR1B P28222 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11007868 0.90 ADRA1D (0.61) CYP2D6CYP1A2CYP3A4CYP2C9ADRA1D
SCHEMBL10744006 0.89 SLC6A4 (0.53) CYP2D6ADRA1DSLC6A4HTR1ADRD2
SCHEMBL10738817 0.85 ADRA1D (0.49) CYP2D6ADRA1DSLC6A4HTR1ADRD2
SCHEMBL11013197 0.83 DRD2 (0.61) CYP2D6CYP1A2CYP3A4CYP2C9ADRA1D
SCHEMBL11047479 0.81 ADRA1D (0.61) CYP2D6ADRA1DSLC6A4HTR2AHTR7
SCHEMBL7649189 0.80 KDM4E (0.67) CYP2D6CYP1A2CYP3A4CYP2C9ADRA1D
SCHEMBL14306777 0.78 ADRA1D (0.80) CYP2D6ADRA1DSLC6A4
SCHEMBL8558927 0.77 ADRA1D (0.63) CYP1A2CYP3A4CYP2C9ADRA1DSLC6A4
Hydrochloric Acid SCHEMBL9031120 0.77 CYP1A2 (0.63) CYP2D6CYP1A2CYP3A4CYP2C9THPO
SCHEMBL8559411 0.76 HTR1A (0.61) CYP2D6CYP1A2CYP3A4CYP2C9THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4665075-A ANTISEROTONINE AGENTS JANSSEN PHARMACEUTICA N.V. (BE) 1987-05-12 US disclosed
EP-0184258-A2 Novel derivatives of hydroxy- or amino-substituted (piperidinylalkyl)quinazolines JANSSEN PHARMACEUTICA N.V. (BE) 1986-06-11 EP disclosed