SCHEMBL7649487

SCHEMBL7649487

CC(C)Oc1ccccc1N1CCN(C(C)c2cccc(C#N)c2)CC1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 5/20 0.45
ADRA1A P35348 5/20 0.45
ADRA1B P35368 5/20 0.45
HTR6 P50406 1/20 0.42
DRD2 P14416 1/20 0.41
UTS2R Q9UKP6 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7645293 0.79 HTR1A (0.50) ADRA1DADRA1AADRA1BDRD2
SCHEMBL8758391 0.79 HTR1A (0.60) ADRA1DADRA1AADRA1BDRD2
SCHEMBL9540921 0.75 HTR1A (0.68) ADRA1DADRA1AADRA1BDRD2
Oxalic Acid SCHEMBL7648371 0.74 HTR1A (0.64) ADRA1DADRA1AADRA1BDRD2
SCHEMBL7690863 0.72 ADRA1A (0.57) ADRA1DADRA1AADRA1B
Bromide SCHEMBL7683252 0.71 ADRA1A (0.56) ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7971839 0.71 DRD4 (0.57) DRD2UTS2R
SCHEMBL14621895 0.70 DRD2 (0.67) ADRA1DADRA1AADRA1BDRD2
SCHEMBL6705579 0.70 ADRA1D (0.47) ADRA1DADRA1AADRA1B
SCHEMBL7301761 0.70 ADRA1A (0.60) ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0563345-B1 NOVEL 4-ARYLPIPERAZINES AND 4-ARYLPIPERIDINES MCNEILAB INC (US) 2002-07-03 EP disclosed
US-5569659-A ANTIPSYCHOTIC AGENT MCNEILAB, INC. (US) 1996-10-29 US disclosed
EP-0563345-A1 NOVEL 4-ARYLPIPERAZINES AND 4-ARYLPIPERIDINES MCNEILAB, INC. (US) 1993-10-06 EP disclosed
WO-1993004682-A1 NOVEL 4-ARYLPIPERAZINES AND 4-ARYLPIPERIDINES MCNEILAB, INC. (US) 1993-03-18 WO disclosed