SCHEMBL7649604

SCHEMBL7649604

CC(C)(C)n1c(=O)c2ccccc2n(CCCCCl)c1=O

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.47
PGR P06401 3/20 0.43
RORA P35398 2/20 0.43
RORC P51449 2/20 0.43
RORB Q92753 2/20 0.43
KDM4E B2RXH2 4/20 0.41
MAPT P10636 1/20 0.41
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 2/20 0.40
HPGD P15428 2/20 0.40
HTT P42858 2/20 0.40
TP53 P04637 1/20 0.40
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656674 0.96 CNR2 (0.46) CNR2PGRRORARORCRORB
SCHEMBL7649598 0.83 TSHR (0.55) CNR2PGRRORARORCRORB
SCHEMBL7649524 0.79 TSHR (0.56) CNR2PGRRORARORCRORB
SCHEMBL5037066 0.77 TNF (0.59) CNR2PGRRORARORCRORB
SCHEMBL31189225 0.76 MPO (0.46) CNR2PGRKDM4EMAPTALDH1A1
SCHEMBL22716908 0.76 MPO (0.46) CNR2PGRKDM4EMAPTALDH1A1
SCHEMBL29179745 0.75 SLC6A4 (0.59) PGRRORARORCRORBMAPT
SCHEMBL4547798 0.74 ERCC1 (0.44) CNR2PGRKDM4EALDH1A1SMN1; SMN2
SCHEMBL4729188 0.74 FABP4 (0.58)
SCHEMBL7657372 0.74 CNR2 (0.57) CNR2KDM4EMAPTSMN1; SMN2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed