SCHEMBL7649901

SCHEMBL7649901

CCN(CC)c1ccc(NC(=O)C(c2ccccc2)N2CCCCC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.60
LMNA P02545 3/20 0.60
TSHR P16473 3/20 0.57
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
NPSR1 Q6W5P4 2/20 0.56
ADRB2 P07550 1/20 0.56
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
NOX1 Q9Y5S8 1/20 0.52
CHRM2 P08172 1/20 0.52
CHRM1 P11229 1/20 0.52
CHRM3 P20309 1/20 0.52
GAA P10253 2/20 0.50
HTT P42858 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7650913 0.99 ALDH1A1 (0.58) ALDH1A1LMNATSHRCYP1A2CYP3A4
SCHEMBL7654548 0.88 ALDH1A1 (0.71) ALDH1A1LMNATSHRCYP1A2CYP3A4
SCHEMBL7649404 0.79 HTR1E (0.70) LMNATSHRCYP1A2CYP3A4CYP2D6
SCHEMBL9912061 0.78 ALDH1A1 (0.66) ALDH1A1LMNATSHRCYP3A4CYP2C19
SCHEMBL14352723 0.78 ALDH1A1 (0.66) ALDH1A1LMNATSHRCYP3A4CYP2C19
SCHEMBL5079881 0.77 ALDH1A1 (0.61) ALDH1A1LMNATSHRCYP3A4CYP2C19
SCHEMBL4901879 0.75 ALDH1A1 (0.58) ALDH1A1LMNATSHRMEN1KMT2A
SCHEMBL2846505 0.73 GAA (0.68) ALDH1A1LMNATSHRCYP1A2CYP3A4
SCHEMBL15354934 0.73 CHRM2 (0.60) ALDH1A1LMNATSHRCYP1A2CYP3A4
SCHEMBL19497139 0.73 CHRM2 (0.60) ALDH1A1LMNATSHRCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407120-B1 ADMINISTERING PYRIDINYLACETAMIDE OR PHENYLACETAMIDE DERIVATIVE TO TREAT CARDIOVASCULAR, EATING, SEXUAL, BRAIN, NERVOUS SYSTEM, GASTROINTESTINAL, UROGENITAL, PSYCHOLOGICAL, AND RESPIRATORY SYSTEM DISORDERS PFIZER INC. 2002-06-18 US disclosed