SCHEMBL7653577

SCHEMBL7653577

O=C(O)CC(NS(=O)(=O)c1ccccc1)N(CC1CC1)C(=O)c1ccc(N2CCN(c3ncccn3)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ITGB3 P05106 3/20 0.40
ITGA2B P08514 3/20 0.40
ITGAV P06756 2/20 0.40
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
GPR119 Q8TDV5 1/20 0.38
ALDH1A1 P00352 4/20 0.37
MAPK1 P28482 3/20 0.37
TSHR P16473 1/20 0.37
APP P05067 1/20 0.37
SMN1; SMN2 Q16637 5/20 0.37
LMNA P02545 4/20 0.37
HTR2A P28223 2/20 0.37
HTR1A P08908 1/20 0.37
LIMK2 P53671 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27475491 0.89 ITGB3 (0.46) ITGB3ITGA2BITGAVALDH1A1MAPK1
SCHEMBL383511 0.89 ITGB3 (0.46) ITGB3ITGA2BITGAVALDH1A1MAPK1
SCHEMBL7649933 0.87 NPC1 (0.43) NPC1RAB9AITGB3ITGA2BITGAV
SCHEMBL7650148 0.86 ITGB3 (0.48) ITGB3ITGA2BITGAVALDH1A1HTR2A
SCHEMBL383369 0.81 ITGB3 (0.64) ITGB3ITGA2BITGAVLIMK2
SCHEMBL7653549 0.81 ITGB3 (0.47) NPC1RAB9AITGB3ITGA2BITGAV
SCHEMBL7651238 0.79 LMNA (0.41) NPC1RAB9AITGB3ITGA2BALDH1A1
SCHEMBL7653506 0.78 NPC1 (0.42) NPC1RAB9AITGB3ITGA2BCA1
SCHEMBL7654428 0.77 ITGB3 (0.48) NPC1RAB9AITGB3ITGA2BITGAV
SCHEMBL7653553 0.75 HTR2A (0.45) NPC1RAB9ACA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed