SCHEMBL7650175

SCHEMBL7650175

O=c1[nH]c(=O)n(CCCCBr)c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.50
HTR1A P08908 1/20 0.50
DRD2 P14416 1/20 0.50
HTR2A P28223 1/20 0.50
DAO P14920 1/20 0.48
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TYMP P19971 1/20 0.43
RAB9A P51151 1/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A2 P23975 1/20 0.43
HRH1 P35367 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10827376 0.95 PARP1 (0.50) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL7298333 0.85 ALDH1A1 (0.55) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL7750879 0.85 PGR (0.55) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL7305582 0.85 HTR1A (0.50) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL7649804 0.84 HTR1A (0.49) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL6295463 0.83 PARP1 (0.50) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL6028786 0.83 PGR (0.60) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL446902 0.83 PARP1 (0.50) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL29528989 0.83 PGR (0.60) PARP1HTR1ADRD2HTR2ADAO
SCHEMBL11009779 0.83 ALDH1A1 (0.60) PARP1HTR1ADRD2HTR2ADAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed