SCHEMBL7650243

SCHEMBL7650243

CCCOc1ccc(F)cc1-c1ccc(C#N)c(=O)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
HPGD P15428 1/20 0.39
BCAT2 O15382 1/20 0.38
BCAT1 P54687 1/20 0.38
PDE5A O76074 3/20 0.37
XDH P47989 1/20 0.37
IDH1 O75874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9702581 0.87 ALDH1A1 (0.44) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7576593 0.87 ALDH1A1 (0.42) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7376004 0.86 PDE5A (0.50) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7644788 0.85 PDE5A (0.45) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7645245 0.85 XDH (0.47) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7647544 0.85 ALDH1A1 (0.54) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7648674 0.84 AR (0.40) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7646410 0.83 ALDH1A1 (0.58) ALDH1A1HPGDXDH
SCHEMBL9851541 0.82 PDE5A (0.51) ALDH1A1KDM4EGLAGAAL3MBTL1
SCHEMBL7648115 0.82 ALDH1A1 (0.46) ALDH1A1KDM4EGLAGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0428268-A2 Pharmaceutical phenylpyridone derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-05-22 EP claimed
US-6479520-B1 REGULATING APOPTOSIS IN HUMAN CELLS WITH COMPOUNDS SUCH AS: 3-CYANO-6-(2-METHOXY-4-METHYLTHIOIPHENYL)-2(1H)-PYRIDINONE CELL PATHWAYS, INC. 2002-11-12 US disclosed
US-6046216-A USEFUL TO INHIBIT THE GROWTH OF NEOPLASTIC CELLS. CELL PATHWAYS, INC. (US) 2000-04-04 US disclosed
EP-0428268-A2 Pharmaceutical phenylpyridone derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-05-22 EP disclosed