SCHEMBL7651811

SCHEMBL7651811

COc1ccc(Cn2c(=O)c3cc([N+](=O)[O-])ccc3n(CCCCBr)c2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.47
TDP2 O95551 1/20 0.47
CNR1 P21554 1/20 0.47
ACHE P22303 1/20 0.47
CNR2 P34972 1/20 0.47
KMT2A Q03164 2/20 0.46
PIK3R1 P27986 1/20 0.46
PIK3CA P42336 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652126 0.92 TDP1 (0.47) TDP1TDP2CNR1ACHECNR2
SCHEMBL7654277 0.85 CCR2 (0.45) KMT2A
SCHEMBL7648500 0.85 HDAC1 (0.45) KMT2A
SCHEMBL7648551 0.82 HDAC1 (0.51)
SCHEMBL7648583 0.81 HDAC1 (0.59) TDP1KMT2A
SCHEMBL7654886 0.81 HDAC1 (0.48)
SCHEMBL7648333 0.79 HDAC6 (0.48) KMT2A
SCHEMBL7656537 0.78 HDAC1 (0.47)
SCHEMBL7651785 0.77 TNF (0.48) TDP1
SCHEMBL7650053 0.76 HDAC1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed