SCHEMBL7652236

SCHEMBL7652236

CCOC(=O)C(C)(C)n1c(=O)[nH]c2ccccc2c1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.55
NPC1 O15118 1/20 0.55
GAA P10253 1/20 0.55
ADORA3 P0DMS8 3/20 0.50
ADORA2A P29274 1/20 0.50
ADORA2B P29275 1/20 0.50
ADORA1 P30542 1/20 0.50
CYP1A2 P05177 1/20 0.50
HSD17B10 Q99714 4/20 0.48
MAPT P10636 3/20 0.48
KDM4E B2RXH2 6/20 0.47
CA12 O43570 1/20 0.47
RNASEH1 O60930 1/20 0.47
ERCC1 P07992 1/20 0.47
ERCC5 P28715 1/20 0.47
FEN1 P39748 1/20 0.47
CA9 Q16790 1/20 0.47
ERCC4 Q92889 1/20 0.47
ALDH1A1 P00352 4/20 0.45
HPGD P15428 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653151 0.85 KDM4E (0.44) SMN1; SMN2NPC1GAAADORA3HSD17B10
SCHEMBL7656051 0.85 ADORA3 (0.50) SMN1; SMN2NPC1GAAADORA3ADORA2A
SCHEMBL7649595 0.85 KDM4E (0.47) SMN1; SMN2NPC1GAAHSD17B10MAPT
SCHEMBL7655615 0.84 SMN1; SMN2 (0.45) SMN1; SMN2NPC1GAAADORA3ADORA2A
SCHEMBL7648344 0.83 CA9 (0.51) GAAHSD17B10KDM4ECA12CA9
SCHEMBL7649684 0.83 CA12 (0.51) SMN1; SMN2CYP1A2HSD17B10MAPTCA12
SCHEMBL7651932 0.83 FEN1 (0.51) SMN1; SMN2MAPTKDM4EFEN1ALDH1A1
SCHEMBL7651842 0.83 CA12 (0.51) SMN1; SMN2NPC1GAAADORA3HSD17B10
SCHEMBL7651738 0.81 SMN1; SMN2 (0.43) SMN1; SMN2NPC1GAAADORA3HSD17B10
SCHEMBL7651882 0.80 ADORA3 (0.54) SMN1; SMN2NPC1GAAADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed