SCHEMBL7651738

SCHEMBL7651738

CCOC(=O)C(C)(C)n1c(=O)[nH]c2ccc(-n3cccc3)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
GAA P10253 1/20 0.43
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
ADORA3 P0DMS8 2/20 0.38
MAPT P10636 4/20 0.37
HSD17B10 Q99714 3/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
HCRTR1 O43613 2/20 0.36
MEN1 O00255 1/20 0.36
RAB9A P51151 1/20 0.36
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
MAT2A P31153 1/20 0.35
JAK2 O60674 1/20 0.34
PAK4 O96013 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7649595 0.84 KDM4E (0.47) SMN1; SMN2NPC1GAAMAPTHSD17B10
SCHEMBL7649684 0.82 CA12 (0.51) SMN1; SMN2CA12CA9MAPTHSD17B10
SCHEMBL7651932 0.82 FEN1 (0.51) SMN1; SMN2MAPTKDM4EALDH1A1KMT2A
SCHEMBL7651842 0.82 CA12 (0.51) SMN1; SMN2NPC1GAACA12CA9
SCHEMBL7652236 0.81 SMN1; SMN2 (0.55) SMN1; SMN2NPC1GAACA12CA9
SCHEMBL7653151 0.80 KDM4E (0.44) SMN1; SMN2NPC1GAAADORA3MAPT
SCHEMBL7657940 0.78 CA12 (0.55) GAACA12CA9MAPTKDM4E
SCHEMBL7651849 0.77 MPO (0.38) SMN1; SMN2NPC1GAAADORA3MAPT
SCHEMBL7648344 0.75 CA9 (0.51) GAACA12CA9HSD17B10KDM4E
SCHEMBL7653115 0.72 SMN1; SMN2 (0.57) SMN1; SMN2NPC1GAAMAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed