SCHEMBL7652330

SCHEMBL7652330

COC(=O)c1cc(C(C)(C)C(=O)OC)ccc1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.50
TDP1 Q9NUW8 2/20 0.47
NPSR1 Q6W5P4 2/20 0.46
ALDH1A1 P00352 4/20 0.45
HPGD P15428 1/20 0.45
VCAM1 P19320 1/20 0.43
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
POLB P06746 1/20 0.42
PDGFRB P09619 1/20 0.41
FGFR1 P11362 1/20 0.41
PDGFRA P16234 1/20 0.41
FLT1 P17948 1/20 0.41
FGFR3 P22607 1/20 0.41
KDR P35968 1/20 0.41
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
MAPK1 P28482 2/20 0.40
GLA P06280 1/20 0.40
CASP3 P42574 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27370615 0.83 CFTR (0.56) SIRT6TDP1ALDH1A1MAPK1MAPT
SCHEMBL4856254 0.82 NPSR1 (0.47) TDP1NPSR1ALDH1A1HPGDVCAM1
SCHEMBL15456899 0.82 CHEK1 (0.49) SIRT6TDP1NPSR1ALDH1A1HPGD
SCHEMBL4854941 0.82 NPSR1 (0.47) SIRT6TDP1NPSR1ALDH1A1HPGD
SCHEMBL18562538 0.81 NPSR1 (0.46) NPSR1ALDH1A1HPGDCNR1CNR2
SCHEMBL6981667 0.79 KMT2A (0.51) TDP1NPSR1ALDH1A1HPGDPOLB
SCHEMBL4857830 0.79 ALDH1A1 (0.49) TDP1NPSR1ALDH1A1HPGDCNR1
SCHEMBL732303 0.79 THRB (0.49) NPSR1ALDH1A1HPGDVCAM1CNR1
SCHEMBL20302045 0.79 NPSR1 (0.47) NPSR1ALDH1A1HPGDVCAM1CNR1
SCHEMBL27868621 0.78 SIRT6 (0.46) SIRT6TDP1NPSR1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed