SCHEMBL7652708

SCHEMBL7652708

CC(C)c1coc(=O)n1-c1cc(F)c(C#N)cc1F

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.38
USP14 P54578 1/20 0.35
BCAT2 O15382 4/20 0.32
BCAT1 P54687 4/20 0.32
PTGS1 P23219 2/20 0.32
PTGS2 P35354 2/20 0.32
PGR P06401 1/20 0.32
AKR1B1 P15121 1/20 0.31
NOTUM Q6P988 1/20 0.31
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23245429 0.68 TRPV4 (0.44) TRPV4USP14BCAT2BCAT1NOTUM
SCHEMBL7653141 0.67 KDM1A (0.33) TRPV4USP14BCAT2BCAT1
SCHEMBL7499656 0.67 BCAT2 (0.41) TRPV4USP14BCAT2BCAT1
SCHEMBL20108199 0.66 DHODH (0.44)
SCHEMBL29816583 0.66 DHODH (0.44)
SCHEMBL6103578 0.66 USP14 (0.38) TRPV4USP14BCAT2BCAT1NOTUM
SCHEMBL7697079 0.64 USP14 (0.37) TRPV4USP14BCAT2BCAT1NOTUM
SCHEMBL12413852 0.64 TRPV4 (0.50) TRPV4PGRAR
SCHEMBL6651303 0.64 TRPV4 (0.71) TRPV4
SCHEMBL8193759 0.63 BCAT2 (0.40) TRPV4USP14BCAT2BCAT1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6395683-B1 CHEMICAL INTERMEDIATE FOR HERBICIDES; APPLYING TO PLANTS BAYER AKTIENGESELLSCHAFT (DE) 2002-05-28 US disclosed
EP-0757673-B1 HETEROCYCLYLBENZONITRILES BAYER AG (DE) 2001-10-04 EP disclosed
US-6100420-A 2-(SULFONYLAMINO OR DERIVATIVE THEREOF),4-AMINO,5-(HALO OR HYDROGEN)BENZONITRILE OF GIVEN FORMULA; CHEMICAL INTERMEDIATE TO CORRESPONDING 4-HETEROCYCLE BENZONITRILE HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2000-08-08 US disclosed
US-5858925-A HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1999-01-12 US disclosed
EP-0757673-A1 HETEROCYCLYLBENZONITRILES BAYER AG (DE) 1997-02-12 EP disclosed
WO-1995029158-A1 HETEROCYCLYLBENZONITRILES BAYER AKTIENGESELLSCHAFT (DE) 1995-11-02 WO disclosed