SCHEMBL7653549

SCHEMBL7653549

O=C(O)[C@H](CN(CC1CC1)C(=O)c1ccc(N2CCN(c3ncccn3)CC2)cc1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.47
ITGA2B P08514 13/20 0.47
ITGAV P06756 8/20 0.46
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MMP3 P08254 1/20 0.40
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
GPR119 Q8TDV5 1/20 0.38
ITGB1 P05556 1/20 0.37
ITGA5 P08648 1/20 0.37
ITGB5 P18084 1/20 0.37
MMP2 P08253 1/20 0.37
MMP13 P45452 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL383510 0.89 ITGB3 (0.53) ITGB3ITGA2BITGAVHTR1AHTR2A
SCHEMBL7649922 0.87 ITGB3 (0.47) ITGB3ITGA2BITGAVHTR1AHTR2A
SCHEMBL7650144 0.86 ITGB3 (0.55) ITGB3ITGA2BITGAVMMP3ITGB1
SCHEMBL383368 0.81 ITGB3 (0.73) ITGB3ITGA2BITGAVMMP3ITGB1
SCHEMBL7653577 0.81 NPC1 (0.41) ITGB3ITGA2BITGAVHTR1AHTR2A
SCHEMBL7653553 0.80 HTR2A (0.45) HTR1AHTR2ANPC1RAB9ACA1
SCHEMBL382418 0.79 ITGB3 (0.43) ITGB3ITGA2BITGAVHTR1AHTR2A
SCHEMBL7651226 0.79 ITGB3 (0.46) ITGB3ITGA2BITGAVMMP2ALDH1A1
SCHEMBL7654405 0.78 ITGB3 (0.74) ITGB3ITGA2BITGAV
SCHEMBL7653489 0.78 ITGB3 (0.46) ITGB3ITGA2BITGAVNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed