SCHEMBL7653706

SCHEMBL7653706

COC(=O)c1ccc(NC(Cn2ccnc2)c2ccc(F)cc2)cc1-c1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.47
CYP51A1 Q16850 5/20 0.45
CYP3A4 P08684 3/20 0.43
CYP2C19 P33261 3/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 2/20 0.43
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CYP26A1 O43174 2/20 0.41
CYP1A2 P05177 1/20 0.41
KDM4E B2RXH2 2/20 0.40
AHR P35869 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
QPCT Q16769 1/20 0.39
SCN9A Q15858 1/20 0.39
NAMPT P43490 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656582 0.89 CYP51A1 (0.49) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7561820 0.84 PTGS2 (0.52) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7656231 0.83 FNTA (0.49) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7662073 0.82 CYP26A1 (0.45) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7568524 0.81 PTGS2 (0.50) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7654320 0.80 FNTA (0.53)
SCHEMBL8211342 0.80 FNTA (0.42) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7657896 0.80 CYP51A1 (0.44) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7669307 0.80 FNTA (0.45) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6
SCHEMBL7656236 0.80 FNTA (0.49) PTGS2CYP51A1CYP3A4CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6410539-B1 ANTICARCINOGENIC AGENTS ASTRAZENCA UK LIMITED (GB) 2002-06-25 US disclosed
EP-1054865-A1 FARNESYL TRANSFERASE INHIBITORS AstraZeneca UK Limited (GB) 2000-11-29 EP disclosed
WO-1999041235-A1 FARNESYL TRANSFERASE INHIBITORS ASTRAZENECA UK LIMITED (GB) 1999-08-19 WO disclosed