SCHEMBL7654891

SCHEMBL7654891

COc1ccc(Cn2c(=O)c3c(C)c(CC(=O)O)ccc3n(CCCCBr)c2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.41
LMNA P02545 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
TSHR P16473 2/20 0.40
CYP2C19 P33261 2/20 0.40
PMP22 Q01453 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RGS12 O14924 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
NFKB1 P19838 1/20 0.40
MAPK1 P28482 1/20 0.40
GNAI1 P63096 1/20 0.40
HIF1A Q16665 1/20 0.40
BLM P54132 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656663 0.77 HDAC1 (0.46) ALDH1A1MEN1KMT2AMAPTHDAC1
SCHEMBL7654886 0.76 HDAC1 (0.48) PTGS2MAPTHDAC1HDAC8HDAC6
SCHEMBL7648500 0.75 HDAC1 (0.45) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL7648551 0.74 HDAC1 (0.51) LMNAALDH1A1MAPTHDAC1HDAC8
SCHEMBL7648583 0.74 HDAC1 (0.59) ALDH1A1MEN1KMT2AMAPTHDAC1
SCHEMBL7654277 0.73 CCR2 (0.45) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL7650053 0.72 HDAC1 (0.52) LMNAALDH1A1MAPTKDM4EHDAC1
SCHEMBL7648333 0.71 HDAC6 (0.48) LMNAALDH1A1MEN1KMT2AMAPT
SCHEMBL7656537 0.71 HDAC1 (0.47) TSHRALDH1A1MAPTHDAC1HDAC8
SCHEMBL7651811 0.70 TDP1 (0.47) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed