SCHEMBL7655428

SCHEMBL7655428

N=C(N)NC1CCN(c2ccc(C(=O)NCCC(=O)ONS(=O)(=O)c3ccccc3)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.44
SMYD3 Q9H7B4 2/20 0.43
ITGB3 P05106 5/20 0.42
ITGA2B P08514 5/20 0.42
ITGAV P06756 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SFRP1 Q8N474 1/20 0.41
CASR P41180 3/20 0.40
TPSAB1 Q15661 1/20 0.40
ADRB3 P13945 1/20 0.40
TGM2 P21980 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462626 0.90 ITGB3 (0.46) SMYD3ITGB3ITGA2BITGAVCASR
SCHEMBL7664584 0.86 CCR5 (0.42) HPGDSSMYD3ITGB3ITGA2BITGAV
SCHEMBL382763 0.84 ITGB3 (0.48) HPGDSITGB3ITGA2BITGAVSFRP1
SCHEMBL382545 0.81 ITGB3 (0.46) HPGDSITGB3ITGA2BITGAVCASR
SCHEMBL382702 0.81 ITGB3 (0.46) HPGDSITGB3ITGA2BITGAVCASR
SCHEMBL7662225 0.80 ITGB3 (0.42) ITGB3ITGA2BITGAVALDH1A1SFRP1
SCHEMBL7658795 0.80 KDM4E (0.55) ITGB3ITGA2BALDH1A1
SCHEMBL7656383 0.80 ITGB3 (0.44) HPGDSITGB3ITGA2BITGAVMEN1
SCHEMBL7651521 0.80 ITGB3 (0.68) ITGB3ITGA2BITGAV
SCHEMBL7654735 0.79 ITGB3 (0.66) HPGDSITGB3ITGA2BITGAVSFRP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420558-B1 COMPOUNDS WITH AMIDINE GROUPS ANTAGONISTIC ACTIVITY, CELL ADHESION INHIBITORY ACTIVITY, HUMAN PLATELET AGGREGATION INHIBITORY ACTIVITY, AND THERAPEUTIC AGENTS MEIJI SEIKA KAISHA, LTD. (JP) 2002-07-16 US claimed
EP-1074543-A1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2001-02-07 EP claimed
US-6420558-B1 COMPOUNDS WITH AMIDINE GROUPS ANTAGONISTIC ACTIVITY, CELL ADHESION INHIBITORY ACTIVITY, HUMAN PLATELET AGGREGATION INHIBITORY ACTIVITY, AND THERAPEUTIC AGENTS MEIJI SEIKA KAISHA, LTD. (JP) 2002-07-16 US disclosed
EP-1074543-A1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2001-02-07 EP disclosed