SCHEMBL7655992

SCHEMBL7655992

O=c1[nH]c2ccccc2c(=O)n1CCOCCO

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.70
HPGD P15428 3/20 0.70
KDM4E B2RXH2 4/20 0.60
HSD17B10 Q99714 3/20 0.58
MAPK1 P28482 1/20 0.58
CYP1A2 P05177 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.55
MPO P05164 2/20 0.53
KMT2A Q03164 2/20 0.53
MEN1 O00255 1/20 0.52
GLA P06280 2/20 0.51
ADORA3 P0DMS8 1/20 0.49
ADORA2A P29274 1/20 0.49
ADORA2B P29275 1/20 0.49
ADORA1 P30542 1/20 0.49
CA12 O43570 1/20 0.49
RNASEH1 O60930 1/20 0.49
ERCC1 P07992 1/20 0.49
ERCC5 P28715 1/20 0.49
FEN1 P39748 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5878601 0.85 ALDH1A1 (0.82) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL7649471 0.84 KDM4E (0.69) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL22716785 0.81 CYP1A2 (0.65) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL31189218 0.81 CYP1A2 (0.65) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL6295502 0.80 ALDH1A1 (0.89) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL7650071 0.79 KDM4E (0.58) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL25335252 0.77 MPO (0.63) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL25333362 0.77 ALDH1A1 (0.64) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL9545441 0.77 ALDH1A1 (0.57) ALDH1A1HPGDKDM4EHSD17B10MAPK1
SCHEMBL8074180 0.76 ALDH1A1 (0.68) ALDH1A1HPGDKDM4EHSD17B10MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed