SCHEMBL765612

SCHEMBL765612

C=C(NCc1ccc(Oc2ccc(Cl)cc2C)cc1)C1(NC(=O)c2cncnc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
PTGER4 P35408 1/20 0.41
LIPG Q9Y5X9 1/20 0.40
HPGD P15428 2/20 0.40
MAPK14 Q16539 3/20 0.39
DDR2 Q16832 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL765842 0.92 BDKRB1 (0.53) BDKRB1SMN1; SMN2CYP3A4CYP1A2CYP2D6
SCHEMBL765624 0.88 MAPK14 (0.53) BDKRB1SMN1; SMN2CYP3A4MAPK14CARM1
SCHEMBL10121140 0.86 BDKRB1 (0.41) BDKRB1SMN1; SMN2CYP3A4PTGER4HPGD
SCHEMBL765546 0.83 BDKRB1 (0.53) BDKRB1SMN1; SMN2CYP3A4PTGER4LIPG
SCHEMBL764501 0.83 BDKRB1 (0.49) BDKRB1CYP3A4PTGER4LIPGMAPK14
SCHEMBL765617 0.83 BDKRB1 (0.52) BDKRB1SMN1; SMN2CYP3A4PTGER4HPGD
SCHEMBL12239078 0.83 BDKRB1 (0.54) BDKRB1SMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL765565 0.82 BDKRB1 (0.56) BDKRB1CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL10121385 0.81 BDKRB1 (0.53) BDKRB1CYP3A4PTGER4LIPGMAPK14
SCHEMBL12238924 0.81 BDKRB1 (0.51) BDKRB1SMN1; SMN2CYP3A4PTGER4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed