SCHEMBL765624

SCHEMBL765624

C=C(NCc1ccc(Oc2ccccc2C)cc1)C1(NC(=O)c2cncnc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.53
BDKRB1 P46663 4/20 0.51
EZH2 Q15910 1/20 0.39
LPAR1 Q92633 3/20 0.38
LPAR5 Q9H1C0 3/20 0.38
CYP3A4 P08684 3/20 0.38
MMP13 P45452 3/20 0.37
HTT P42858 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
EGLN1 Q9GZT9 1/20 0.37
MMP2 P08253 1/20 0.36
STAT3 P40763 1/20 0.36
CARM1 Q86X55 1/20 0.36
PRMT6 Q96LA8 1/20 0.36
NOTUM Q6P988 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL764461 0.92 BDKRB1 (0.61) MAPK14BDKRB1EZH2LPAR1LPAR5
SCHEMBL765612 0.88 BDKRB1 (0.45) MAPK14BDKRB1CYP3A4HTTSMN1; SMN2
SCHEMBL10121101 0.86 BDKRB1 (0.45) MAPK14BDKRB1CYP3A4HTTSMN1; SMN2
SCHEMBL764458 0.82 BDKRB1 (0.64) MAPK14BDKRB1EZH2CYP3A4LMNA
SCHEMBL10121331 0.81 BDKRB1 (0.60) MAPK14BDKRB1CYP3A4MMP13HTT
SCHEMBL764501 0.81 BDKRB1 (0.49) MAPK14BDKRB1CYP3A4LMNA
SCHEMBL10121385 0.81 BDKRB1 (0.53) MAPK14BDKRB1CYP3A4CARM1PRMT6
SCHEMBL12239067 0.81 BDKRB1 (0.60) MAPK14BDKRB1CYP3A4MMP13HTT
SCHEMBL12239078 0.80 BDKRB1 (0.54) MAPK14BDKRB1CYP3A4MMP13HTT
SCHEMBL765172 0.80 BDKRB1 (0.58) MAPK14BDKRB1CYP3A4MMP13HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed