SCHEMBL765653

SCHEMBL765653

O=S(=O)(c1ccc(Cl)cc1)C1CCCCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
MAPK1 P28482 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CYP3A4 P08684 1/20 0.46
GAA P10253 1/20 0.46
PSEN1 P49768 5/20 0.46
PSEN2 P49810 5/20 0.46
APH1B Q8WW43 5/20 0.46
NCSTN Q92542 5/20 0.46
APH1A Q96BI3 5/20 0.46
PSENEN Q9NZ42 5/20 0.46
ACHE P22303 1/20 0.46
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
CTSG P08311 1/20 0.44
CMA1 P23946 1/20 0.44
CNR1 P21554 1/20 0.44
DRD2 P14416 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL217625 0.98 ALDH1A1 (0.48) ALDH1A1MAPK1MEN1KMT2ACYP3A4
SCHEMBL31518328 0.84 NAMPT (0.45) ALDH1A1CYP2C9HTR2AGSRTXNRD1
SCHEMBL4674685 0.81 ALDH1A1 (0.43) ALDH1A1MAPK1MEN1KMT2ACYP3A4
SCHEMBL2798239 0.81 MAPT (0.50) ALDH1A1MAPK1CYP3A4PSEN1PSEN2
SCHEMBL25296150 0.80 MAPK1 (0.56) ALDH1A1MAPK1GAACA12CA2
SCHEMBL20379865 0.80 TSHR (0.46) ALDH1A1MEN1KMT2ACYP3A4GAA
SCHEMBL11507747 0.80 ALDH1A1 (0.56) ALDH1A1KMT2ACYP3A4GAAACHE
SCHEMBL31518353 0.80 LMNA (0.45) ALDH1A1MAPK1CYP2C9CYP2C19HTR2A
SCHEMBL23633178 0.80 MMP13 (0.44) CYP2C9HTR2AGSRTXNRD1
SCHEMBL9576066 0.80 ESR1 (0.47) KMT2ACYP2C9CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888050-B1 cis-4-[(4-chlorophenyl)sulfonyl]-4-(2,5-difluorophenyl)cyclohexanepropanoic acid for the treatment of cancer MERCK SHARP & DOHME (GB) 2012-03-21 EP disclosed